Azaserine

Azaserine

SCHEMBL8861

[N-]=[N+]=CC(=O)OC[C@H](N)C(=O)O

nearest known ligand 0.38

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC1A5 Q15758 1/20 0.38
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37
NOS2 P35228 1/20 0.37
IDO1 P14902 2/20 0.36
PTGS1 P23219 1/20 0.34
SLC7A11 Q9UPY5 1/20 0.34
GFPT1 Q06210 1/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
GRIK1 P39086 6/20 0.32
GRIK2 Q13002 5/20 0.32
GSR P00390 2/20 0.32
SLC1A1 P43005 2/20 0.32
GRM1 Q13255 2/20 0.32
GRM2 Q14416 2/20 0.32
GRIA2 P42262 2/20 0.32
GRIA4 P48058 2/20 0.32
GRIK3 Q13003 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Azaserine SCHEMBL8862 1.00 SLC1A5 (0.38) SLC1A5NOS3NOS1NOS2IDO1
Azaserine SCHEMBL487222 1.00 SLC1A5 (0.38) SLC1A5NOS3NOS1NOS2IDO1
Azaserine SCHEMBL3312110 1.00 SLC1A5 (0.38) SLC1A5NOS3NOS1NOS2IDO1
Azaserine SCHEMBL27500218 0.98 SLC1A5 (0.37) SLC1A5NOS3NOS1NOS2IDO1
Azaserine SCHEMBL607082 0.98 SLC1A5 (0.37) SLC1A5NOS3NOS1NOS2IDO1
SCHEMBL607081 0.84
Azaserine SCHEMBL6824548 0.82 ALOX15 (0.47) NOS3NOS1NOS2CYP1A2GRIK1
SCHEMBL31237462 0.81 IDO1 (0.40) SLC1A5NOS3NOS1NOS2IDO1
SCHEMBL26934495 0.81 IDO1 (0.40) SLC1A5NOS3NOS1NOS2IDO1
Azaserine SCHEMBL81760 0.78 ALDH1A1 (0.41) SLC1A5IDO1SLC7A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 31931 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4748859-A2 CHEMICALLY AND PHOTOCHEMICALLY INITIATED CELL MEMBRANE BLEBBING TO INDUCE CELL VESICLE PRODUCTION, MODIFICATIONS THEREOF, AND USES THEREOF The Regents of the University of California (US) 2026-05-27 EP claimed
US-20260137794-A1 LIGAND-DRUG CONJUGATE AND USE THEREOF SYSTIMMUNE INC (US) 2026-05-21 US claimed
EP-4743490-A1 HUMANIZED ANTI-CD7 ANTIBODY Christian-Albrechts-Universität zu Kiel (DE) 2026-05-20 EP claimed
WO-2026099502-A1 NOVEL DRUG CONJUGATES FOR TESTING CELLULAR DRUG UPTAKE Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2026-05-15 WO claimed
US-20260115305-A1 LINKERS, CONJUGATES AND APPLICATIONS THEREOF GENEQUANTUM HEALTHCARE SUZHOU CO LTD (CN) 2026-04-30 US claimed
US-20260108619-A1 CONJUGATION LINKERS, CELL BINDING MOLECULE-DRUG CONJUGATES CONTAINING THE LINKERS, METHODS OF MAKING AND USES SUCH CONJUGATES WITH THE LINKERS HANGZHOU DAC BIOTECH CO., LTD. (CN) 2026-04-23 US claimed
US-20260085100-A1 METHODS OF ANTIGEN PRODUCTION THE WISTAR INSTITUTE OF ANATOMY AND BIOLOGY (US) 2026-03-26 US claimed
US-20260077056-A1 LINKER-PAYLOAD COMPOUND, CONJUGATES AND APPLICATIONS THEREOF GENEQUANTUM HEALTHCARE SUZHOU CO LTD (CN) 2026-03-19 US claimed
US-12576124-B2 Formulation of a conjugate of a tubulysin analog to a cell-binding molecule HANGZHOU DAC BIOTECH CO., LTD (CN) 2026-03-17 US claimed
EP-4698185-A1 METHODS AND SYSTEMS FOR IMPROVING ANTI-CANCER THERAPIES Osasuna Therapeutics SA (CH) 2026-02-25 EP claimed
EP-0081107-B1 PROCESS FOR PRODUCING L-TRYPTOPHAN BY FERMENTATION AJINOMOTO CO., INC. (JP) 1986-09-10 EP claimed
US-4601982-A Method for producing L-tryptophan by fermentation with a brevibacterium flavum mutant AJINOMOTO COMPANY INCORPORATED (JP) 1986-07-22 US claimed
EP-0105360-A4 ANTIBODIES HAVING DUAL SPECIFICITIES, THEIR PREPARATION AND USES THEREFOR. HYBRITECH INC (US) 1986-07-08 EP claimed
EP-0183006-A2 A recombinant DNA-molecule, coryneform bacteria carrying recombinant DNA and process for producing an aromatic amino acid by using the same AJINOMOTO CO., INC. (JP) 1986-06-04 EP claimed
US-4560652-A BACILLUS MUTANT AZASERINE, METHYL-TRYPTOPHAN AND FLUORO-TRYPTOPHAN RESISTANT; FEEDS AJINOMOTO CO., INC. (JP) 1985-12-24 US claimed
EP-0160550-A2 Human lymphoblastoid cell line and hybridomas derived therefrom and antibodies produced from such hybridomas, and the production and use of the aforesaid CETUS CORPORATION (US) 1985-11-06 EP claimed
EP-0118917-A2 Method for production of biologically active substances Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1984-09-19 EP claimed
EP-0105360-A1 ANTIBODIES HAVING DUAL SPECIFICITIES, THEIR PREPARATION AND USES THEREFOR HYBRITECH INCORPORATED (US) 1984-04-18 EP claimed
WO-1983003679-A1 ANTIBODIES HAVING DUAL SPECIFICITIES, THEIR PREPARATION AND USES THEREFOR HYBRITECH INC (US) 1983-10-27 WO claimed
EP-0081107-A2 Process for producing L-tryptophan by fermentation AJINOMOTO CO., INC. (JP) 1983-06-15 EP claimed