SCHEMBL8863522

SCHEMBL8863522

O=C1c2ccc(F)cc2C(=O)N1CCN1CCC(c2onc3cc(F)ccc23)CC1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.46
DRD2 P14416 12/20 0.43
SLC6A4 P31645 1/20 0.43
HTR2A P28223 5/20 0.43
HTR1A P08908 4/20 0.43
HTR7 P34969 1/20 0.41
DRD3 P35462 1/20 0.41
HTR6 P50406 1/20 0.41
KCNH2 Q12809 1/20 0.41
HTR2C P28335 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8787429 0.94 DRD2 (0.47) ACHEDRD2SLC6A4HTR2AHTR1A
SCHEMBL8789177 0.93 ACHE (0.42) ACHEDRD2SLC6A4HTR2AHTR1A
SCHEMBL7355692 0.93 ACHE (0.42) ACHEDRD2SLC6A4HTR2AHTR1A
Hydrochloric Acid SCHEMBL8787530 0.93 DRD2 (0.46) ACHEDRD2SLC6A4HTR2AHTR1A
SCHEMBL9096725 0.92 ACHE (0.44) ACHEDRD2SLC6A4HTR2AHTR1A
SCHEMBL7773189 0.91 DRD2 (0.46) ACHEDRD2SLC6A4HTR2AHTR1A
SCHEMBL8787639 0.91 ACHE (0.41) ACHEDRD2SLC6A4HTR2AHTR1A
SCHEMBL8787558 0.88 DRD2 (0.49) DRD2HTR2AHTR1AKCNH2
SCHEMBL8788723 0.88 DRD2 (0.49) DRD2SLC6A4HTR2AHTR1AHTR7
SCHEMBL8789443 0.88 ACHE (0.46) ACHEDRD2SLC6A4HTR2AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5637710-A ETHYL 3-(4-(6-FLUORO-1,2-BENZISOTHIAZOLE-3-YL)-1-PIPERIDINYL)PROPIO -NATE; ETHYL 3-(4-(6-FLUORO-1H-INDAZOLE-3-YL)-1-PIPERAZINYL) PROPIONATE HOECHST MARION ROUSSEL, INC. (US) 1997-06-10 US disclosed
US-5561128-A ANALGESICS; ANTIPSYCHOTIC AGENTS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1996-10-01 US disclosed