SCHEMBL8787429

SCHEMBL8787429

O=C1c2ccccc2C(=O)N1CCN1CCC(c2onc3cc(F)ccc23)CC1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 9/20 0.47
HTR2A P28223 7/20 0.47
HTR1A P08908 5/20 0.47
ACHE P22303 2/20 0.46
HTR2C P28335 1/20 0.43
SLC6A4 P31645 1/20 0.43
MCHR1 Q99705 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8787530 0.99 DRD2 (0.46) DRD2HTR2AHTR1AACHEHTR2C
SCHEMBL8787558 0.94 DRD2 (0.49) DRD2HTR2AHTR1AMCHR1
SCHEMBL8788723 0.94 DRD2 (0.49) DRD2HTR2AHTR1AHTR2CSLC6A4
SCHEMBL8863522 0.94 ACHE (0.46) DRD2HTR2AHTR1AACHEHTR2C
SCHEMBL9096725 0.90 ACHE (0.44) DRD2HTR2AHTR1AACHESLC6A4
SCHEMBL7355692 0.89 ACHE (0.42) DRD2HTR2AHTR1AACHEHTR2C
SCHEMBL8789177 0.89 ACHE (0.42) DRD2HTR2AHTR1AACHEHTR2C
SCHEMBL8789443 0.88 ACHE (0.46) DRD2HTR2AHTR1AACHESLC6A4
SCHEMBL8788754 0.87 DRD2 (0.41) DRD2HTR2AHTR1AACHEHTR2C
SCHEMBL7773189 0.87 DRD2 (0.46) DRD2HTR2AHTR1AACHEHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0730452-A4 HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES AND THEIR USE AS ANTIPSYCHOTICS AND ANALGETICS HOECHST ROUSSEL PHARMA (US) 1997-03-19 EP claimed
EP-0730452-A1 HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES AND THEIR USE AS ANTIPSYCHOTICS AND ANALGETICS HOECHST MARION ROUSSEL, Inc. (US) 1996-09-11 EP claimed
EP-0730452-A4 HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES AND THEIR USE AS ANTIPSYCHOTICS AND ANALGETICS HOECHST ROUSSEL PHARMA (US) 1997-03-19 EP disclosed
EP-0730452-A1 HETEROARYLPIPERIDINES, PYRROLIDINES AND PIPERAZINES AND THEIR USE AS ANTIPSYCHOTICS AND ANALGETICS HOECHST MARION ROUSSEL, Inc. (US) 1996-09-11 EP disclosed