SCHEMBL8864262

SCHEMBL8864262

CCCCOc1ccc(O)cc1C

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 11/20 0.59
LTA4H P09960 2/20 0.50
NR5A1 Q13285 1/20 0.50
MEN1 O00255 1/20 0.47
NPC1 O15118 1/20 0.47
ALDH1A1 P00352 1/20 0.47
GAA P10253 1/20 0.47
MAPT P10636 1/20 0.47
RAB9A P51151 1/20 0.47
KMT2A Q03164 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
THRA P10827 1/20 0.46
THRB P10828 1/20 0.46
WDR5 P61964 2/20 0.45
CYSLTR2 Q9NS75 1/20 0.43
CYSLTR1 Q9Y271 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11071449 0.95 ESR1 (0.58) ESR1LTA4HNR5A1THRATHRB
SCHEMBL9699080 0.93 ESR1 (0.61) ESR1LTA4HNR5A1MEN1MAPT
SCHEMBL11796987 0.93 ESR1 (0.61) ESR1LTA4HNR5A1MEN1MAPT
SCHEMBL9697402 0.93 ESR1 (0.61) ESR1LTA4HNR5A1MEN1MAPT
SCHEMBL9699688 0.93 ESR1 (0.61) ESR1LTA4HNR5A1MEN1MAPT
SCHEMBL14747883 0.91 ESR1 (0.49) ESR1LTA4HMEN1ALDH1A1GAA
SCHEMBL3291614 0.86 ESR1 (0.54) ESR1LTA4HNR5A1THRATHRB
SCHEMBL3995606 0.85 LTA4H (0.50) ESR1LTA4HNR5A1MEN1NPC1
SCHEMBL3006259 0.83 ALDH1A1 (0.60) ESR1LTA4HNR5A1MEN1NPC1
SCHEMBL19433121 0.83 LTA4H (0.52) ESR1LTA4HNR5A1MEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0887346-B1 N-Phenyl-alkylsulfonamide derivatives, their preparation and their use as alpha1A/1L adrenoceptor agonists HOFFMANN LA ROCHE (CH) 2007-12-12 EP disclosed
CN-1059895-C Method for preparing alkoxy substituted triphenylamine MITSUI TOATSU CHEMICALS (JP) 2000-12-27 CN disclosed
US-5654483-A REACTING ALKOXY-SUBSTITUTED CYCLOHEXANONE WITH DIPHENYLAMINE WHILE FORMING CYCLOHEXANONE FROM ALKOXY-SUBSTITUTED PHENOL IN PRESENCE OF SURFACE-SUPPORTED HYDROGEN TRANSFER CATALYST MITSUI TOATSU CHEMICALS, INC. (JP) 1997-08-05 US disclosed
CN-1130174-A Method for preparing alkoxy substituted triphenylamine MITSUI TOATSU CHEMICALS (JP) 1996-09-04 CN disclosed