SCHEMBL8864636

SCHEMBL8864636

Cn1nc(-c2ccc([N+](=O)[O-])cc2)c2ccccc2c1=O

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.60
L3MBTL1 Q9Y468 2/20 0.58
ALDH1A1 P00352 5/20 0.56
SMN1; SMN2 Q16637 3/20 0.56
MAPT P10636 5/20 0.56
POLB P06746 2/20 0.56
LMNA P02545 1/20 0.56
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
ENPP1 P22413 2/20 0.53
NPC1 O15118 2/20 0.52
RAB9A P51151 1/20 0.52
HTT P42858 2/20 0.52
GAA P10253 1/20 0.52
MAPK1 P28482 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20379747 0.84 L3MBTL1 (0.71) L3MBTL1ALDH1A1SMN1; SMN2MAPTLMNA
SCHEMBL8224982 0.81 HPGD (0.74) HPGDL3MBTL1ALDH1A1SMN1; SMN2MAPT
SCHEMBL8864677 0.80 HPGD (0.70) HPGDL3MBTL1ALDH1A1SMN1; SMN2MAPT
SCHEMBL1376771 0.79 HPGD (0.71) HPGDL3MBTL1ALDH1A1SMN1; SMN2MAPT
SCHEMBL29382447 0.79 SMN1; SMN2 (0.70) HPGDL3MBTL1ALDH1A1SMN1; SMN2MAPT
SCHEMBL8865071 0.79 HPGD (0.67) HPGDL3MBTL1ALDH1A1SMN1; SMN2MAPT
SCHEMBL8864626 0.79 HPGD (0.67) HPGDL3MBTL1ALDH1A1SMN1; SMN2MAPT
SCHEMBL8864802 0.79 HPGD (0.67) HPGDL3MBTL1ALDH1A1SMN1; SMN2MAPT
SCHEMBL8864565 0.78 ALOX5 (0.66) HPGDL3MBTL1ALDH1A1SMN1; SMN2MAPT
SCHEMBL8268002 0.77 HPGD (0.64) HPGDL3MBTL1ALDH1A1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5624922-A Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC. (US) 1997-04-29 US disclosed
EP-0597540-B1 Aryl-fused and hetaryl-fused-2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC (US) 1996-06-05 EP disclosed
US-5380721-A Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC. (US) 1995-01-10 US disclosed
EP-0597540-A1 Aryl-fused and hetaryl-fused-2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC. (US) 1994-05-18 EP disclosed