SCHEMBL8865160

SCHEMBL8865160

CC(=O)Oc1ccc(C#Cc2cc3c(cc2C)SC(C)(C)CC3(C)C)nc1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.37
RARA P10276 2/20 0.37
RARB P10826 2/20 0.37
RARG P13631 2/20 0.37
KMT2A Q03164 1/20 0.37
CYP26A1 O43174 1/20 0.36
ALDH1A1 P00352 1/20 0.33
F2 P00734 1/20 0.33
GLA P06280 1/20 0.33
HPGD P15428 1/20 0.33
ACACB O00763 4/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8865251 0.90 CYP3A4 (0.39) CYP3A4RARARARBRARGKMT2A
SCHEMBL8865583 0.85 ALOX5 (0.38) CYP3A4RARARARBRARGKMT2A
SCHEMBL8865464 0.84 CYP3A4 (0.49) CYP3A4RARARARBRARGKMT2A
SCHEMBL8890100 0.83 CYP3A4 (0.52) CYP3A4RARARARBRARGKMT2A
SCHEMBL8865150 0.81 RARA (0.58) CYP3A4RARARARBRARGKMT2A
SCHEMBL8874466 0.81 CYP26A1 (0.38) CYP3A4RARARARBRARGKMT2A
SCHEMBL8875274 0.78 CYP3A4 (0.41) CYP3A4RARARARBRARGKMT2A
SCHEMBL8661571 0.77 CYP3A4 (0.43) CYP3A4RARARARBRARGKMT2A
SCHEMBL8875128 0.76 CYP3A4 (0.40) CYP3A4RARARARBRARGKMT2A
SCHEMBL8865783 0.76 RARA (0.33) CYP3A4RARARARBRARGKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5677323-A SKIN DISORDERS, PSORIASIS ALLERGAN (US) 1997-10-14 US disclosed