SCHEMBL8890100

SCHEMBL8890100

Cc1cc2c(cc1C#Cc1ccc(C(=O)O)cn1)C(C)(C)CC(C)(C)S2

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.52
CYP26A1 O43174 2/20 0.52
RARB P10826 8/20 0.42
RARG P13631 8/20 0.42
RARA P10276 7/20 0.42
KMT2A Q03164 1/20 0.42
RXRA P19793 9/20 0.40
RXRB P28702 7/20 0.40
RXRG P48443 7/20 0.40
PPARG P37231 1/20 0.39
SLC16A3 O15427 1/20 0.36
CRABP2 P29373 1/20 0.34
GRM5 P41594 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8865150 0.88 RARA (0.58) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL8874466 0.85 CYP26A1 (0.38) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL9180876 0.84 RARB (0.51) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL6664628 0.84 CYP3A4 (0.71) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL8892530 0.83 CYP3A4 (0.71) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL8865160 0.83 CYP3A4 (0.37) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL9318320 0.82 RXRA (0.58) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL8875070 0.80 CYP3A4 (0.32) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL8865484 0.80 RARA (0.58) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL8891765 0.80 CYP3A4 (0.46) CYP3A4CYP26A1RARBRARGRARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5616597-A ANTIACNE, ANTIPSORIASIS COMPOUNDS ALLERGAN (US) 1997-04-01 US disclosed
US-5272156-A Acetylenes disubstituted with a heteroaromatic group and a 2-substituted 1,2,3,4-tetrahydroquinolinyl group having retinoid-like activity ALLERGAN, INC. (US) 1993-12-21 US disclosed
US-5183827-A Skin disorders ALLERGAN, INC. (US) 1993-02-02 US disclosed
US-5045551-A Acetylenes disubstituted with a heteroaromatic group and a 2-substituted chromanyl, thiochromanyl or 1,2,3,4-tetrahydroquinolinyl group having retinoid-like activity ALLERGAN, INC. (US) 1991-09-03 US disclosed