SCHEMBL8866735

SCHEMBL8866735

CC(Cc1ccccc1)(NC(=O)CN)c1ccc(OC(=O)/C=C\C(=O)Oc2ccc(C(C)(Cc3ccccc3)NC(=O)CN)cc2)cc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.72
CYP1A2 P05177 1/20 0.72
RECQL P46063 1/20 0.72
MAPK1 P28482 1/20 0.70
GAA P10253 3/20 0.40
CYP2C19 P33261 2/20 0.40
POLB P06746 1/20 0.40
LTA4H P09960 1/20 0.40
KMT2A Q03164 5/20 0.39
MEN1 O00255 4/20 0.39
ALDH1A1 P00352 2/20 0.39
LMNA P02545 2/20 0.39
MAPT P10636 3/20 0.39
KDM4E B2RXH2 2/20 0.39
CYP2C9 P11712 1/20 0.39
TSHR P16473 1/20 0.37
MITF O75030 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
RAB9A P51151 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8866359 0.95 CYP3A4 (0.72) CYP3A4CYP1A2RECQLMAPK1GAA
SCHEMBL9053526 0.86 CYP1A2 (0.78) CYP3A4CYP1A2RECQLMAPK1GAA
Maleic Acid SCHEMBL8865839 0.86 CYP1A2 (0.69) CYP3A4CYP1A2RECQLMAPK1GAA
Fumaric Acid SCHEMBL8865851 0.86 CYP1A2 (0.69) CYP3A4CYP1A2RECQLMAPK1GAA
Remacemide SCHEMBL20769836 0.85 CYP1A2 (1.00) CYP3A4CYP1A2RECQLMAPK1CYP2C19
Remacemide SCHEMBL151148 0.85 CYP1A2 (1.00) CYP3A4CYP1A2RECQLMAPK1CYP2C19
Remacemide SCHEMBL7266326 0.84 CYP3A4 (0.86) CYP3A4CYP1A2RECQLMAPK1CYP2C19
Remacemide SCHEMBL31270066 0.84 CYP3A4 (0.86) CYP3A4CYP1A2RECQLMAPK1CYP2C19
Remacemide SCHEMBL7266094 0.84 CYP3A4 (0.86) CYP3A4CYP1A2RECQLMAPK1CYP2C19
Remacemide SCHEMBL635940 0.83 MAPK1 (1.00) CYP3A4CYP1A2RECQLMAPK1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5605916-A Arylalkyl-amines having anticonvulsant and neuroprotective properties ASTRA AB (SE) 1997-02-25 US disclosed
US-5539120-A Arylalkyl-amines having anticonvulsant and neuroprotective properties AGENCE SPATIALE EUROPEENNE (FR) 1996-07-23 US disclosed
EP-0356035-B1 Arylkalkyl-amines and -amides having anticonvulsant and neuroprotective properties ASTRA AB (SE) 1996-03-13 EP disclosed
US-5430044-A Arylalkyl-amines and -amides having anticonvulsant and neuroprotective properties FISONS CORPORATION (GB) 1995-07-04 US disclosed
EP-0648489-A1 Arylalkylamides having neuroprotective properties FISONS CORPORATION (US) 1995-04-19 EP disclosed
EP-0648745-A1 Arylalkylamine having anticonvulsant and neuroprotective properties Astra Aktiebolag (SE) 1995-04-19 EP disclosed
US-5331007-A Arylalkyl-amines and -amides having anticonvulsant and neuroprotective properties FISONS CORPORATION (US) 1994-07-19 US disclosed
WO-1991011995-A1 ARYLALKYL-AMINES AND -AMIDES HAVING ANTICONVULSANT AND NEUROPROTECTIVE PROPERTIES FISONS CORPORATION (US) 1991-08-22 WO disclosed
EP-0356035-A2 Arylkalkyl-amines and -amides having anticonvulsant and neuroprotective properties Astra Aktiebolag (SE) 1990-02-28 EP disclosed