SCHEMBL9053526

SCHEMBL9053526

COc1ccc(C(C)(Cc2ccccc2)NC(=O)CN)cc1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.78
CYP3A4 P08684 2/20 0.78
RECQL P46063 2/20 0.78
MAPK1 P28482 2/20 0.76
RAB9A P51151 3/20 0.47
NPC1 O15118 3/20 0.47
MMP1 P03956 2/20 0.46
MMP13 P45452 2/20 0.46
MMP9 P14780 1/20 0.46
PLAU P00749 1/20 0.46
ELANE P08246 1/20 0.46
ALDH1A1 P00352 5/20 0.46
MAPT P10636 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
TSHR P16473 1/20 0.45
KIF11 P52732 1/20 0.44
CNR2 P34972 1/20 0.44
LMNA P02545 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5304269 0.95 CYP1A2 (0.78) CYP1A2CYP3A4RECQLMAPK1RAB9A
Fumaric Acid SCHEMBL8865851 0.94 CYP1A2 (0.69) CYP1A2CYP3A4RECQLMAPK1RAB9A
Maleic Acid SCHEMBL8865839 0.94 CYP1A2 (0.69) CYP1A2CYP3A4RECQLMAPK1RAB9A
Maleic Acid SCHEMBL8866481 0.89 CYP1A2 (0.69) CYP1A2CYP3A4RECQLMAPK1RAB9A
Fumaric Acid SCHEMBL8866493 0.89 CYP1A2 (0.69) CYP1A2CYP3A4RECQLMAPK1RAB9A
Remacemide SCHEMBL20769836 0.88 CYP1A2 (1.00) CYP1A2CYP3A4RECQLMAPK1ALDH1A1
Remacemide SCHEMBL151148 0.88 CYP1A2 (1.00) CYP1A2CYP3A4RECQLMAPK1ALDH1A1
SCHEMBL5306970 0.86 CYP1A2 (0.72) CYP1A2CYP3A4RECQLMAPK1RAB9A
SCHEMBL8866735 0.86 CYP3A4 (0.72) CYP1A2CYP3A4RECQLMAPK1RAB9A
Remacemide SCHEMBL635940 0.86 MAPK1 (1.00) CYP1A2CYP3A4RECQLMAPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0356035-B1 Arylkalkyl-amines and -amides having anticonvulsant and neuroprotective properties ASTRA AB (SE) 1996-03-13 EP claimed
WO-1991011995-A1 ARYLALKYL-AMINES AND -AMIDES HAVING ANTICONVULSANT AND NEUROPROTECTIVE PROPERTIES FISONS CORPORATION (US) 1991-08-22 WO claimed
EP-0356035-A2 Arylkalkyl-amines and -amides having anticonvulsant and neuroprotective properties Astra Aktiebolag (SE) 1990-02-28 EP claimed