SCHEMBL8867093

SCHEMBL8867093

CCOC(=O)c1sc(-c2ccc(O)c(Cl)c2)nc1C

nearest known ligand 0.63

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 8/20 0.62
DBF4 Q9UBU7 8/20 0.62
TRPM8 Q7Z2W7 6/20 0.59
MAPT P10636 4/20 0.59
KDM4E B2RXH2 3/20 0.53
ALDH1A1 P00352 1/20 0.53
LMNA P02545 1/20 0.52
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
HSP90AA1 P07900 1/20 0.50
CRHBP P24387 1/20 0.50
CRHR2 Q13324 1/20 0.50
DHODH Q02127 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12186978 0.88 CDC7 (0.64) CDC7DBF4TRPM8MAPTKDM4E
SCHEMBL8867336 0.86 CDC7 (0.62) CDC7DBF4TRPM8MAPTKDM4E
SCHEMBL19523297 0.85 CDC7 (0.62) CDC7DBF4TRPM8MAPTKDM4E
SCHEMBL455876 0.85 CDC7 (0.62) CDC7DBF4TRPM8MAPTKDM4E
SCHEMBL15383553 0.84 ALDH1A1 (0.62) CDC7DBF4TRPM8MAPTKDM4E
SCHEMBL29627451 0.83 CDC7 (0.59) CDC7DBF4TRPM8MAPTKDM4E
SCHEMBL454793 0.83 CDC7 (0.59) CDC7DBF4TRPM8MAPTKDM4E
SCHEMBL2885708 0.83 TRPM8 (0.78) CDC7DBF4TRPM8MAPTKDM4E
SCHEMBL19523327 0.82 MAPT (0.58) CDC7DBF4TRPM8MAPTKDM4E
SCHEMBL30804867 0.82 CDC7 (0.58) CDC7DBF4TRPM8MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2927219-B1 2-ARYL SELENAZOLE COMPOUND AND PHARMACEUTICAL COMPOSITION THEREOF ATOM BIOSCIENCE AND PHARMACEUTICAL CO LTD (CN) 2018-05-30 EP disclosed
US-9802907-B2 2-aryl selenazole compound and pharmaceutical composition thereof JIANGSU ATOM BIOSCIENCE AND PHARMACEUTICAL CO., LTD. (CN) 2017-10-31 US disclosed
US-5614520-A 2-arylthiazole derivatives and pharmaceutical composition thereof TEIJIN LIMITED (JP) 1997-03-25 US disclosed
EP-0513379-B1 2-ARYLTHIAZOLE DERIVATIVE AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME TEIJIN LTD (JP) 1996-09-11 EP disclosed
EP-0513379-A1 2-ARYLTHIAZOLE DERIVATIVE AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME TEIJIN LIMITED (JP) 1992-11-19 EP disclosed