SCHEMBL8867115

SCHEMBL8867115

Cc1nc(-c2ccc(C(=O)c3ccccc3)cc2)sc1C(=O)O

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 8/20 0.77
RAB9A P51151 8/20 0.70
KDM4E B2RXH2 4/20 0.70
GAA P10253 2/20 0.70
NPC1 O15118 5/20 0.67
POLB P06746 1/20 0.67
KMT2A Q03164 3/20 0.59
ALDH1A1 P00352 7/20 0.58
HPGD P15428 3/20 0.58
NPSR1 Q6W5P4 1/20 0.58
XDH P47989 1/20 0.58
MAPT P10636 4/20 0.56
TARBP2 Q15633 1/20 0.55
RARA P10276 1/20 0.52
RARB P10826 1/20 0.52
RARG P13631 1/20 0.52
LMNA P02545 1/20 0.52
ATM Q13315 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.51
MEN1 O00255 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8868807 0.91 RAB9A (0.85) SMN1; SMN2RAB9AKDM4EGAANPC1
SCHEMBL289112 0.88 SMN1; SMN2 (0.93) SMN1; SMN2RAB9AKDM4EGAANPC1
SCHEMBL8867051 0.88 RAB9A (0.79) SMN1; SMN2RAB9AKDM4EGAANPC1
SCHEMBL1327631 0.88 SMN1; SMN2 (1.00) SMN1; SMN2RAB9AKDM4EGAANPC1
SCHEMBL8866740 0.87 SMN1; SMN2 (0.71) SMN1; SMN2RAB9AKDM4EGAANPC1
SCHEMBL8867673 0.84 CDC7 (0.67) SMN1; SMN2RAB9AKDM4EGAANPC1
SCHEMBL892234 0.83 RAB9A (1.00) SMN1; SMN2RAB9AKDM4EGAANPC1
SCHEMBL8868197 0.82 RAB9A (0.70) SMN1; SMN2RAB9AKDM4EGAANPC1
SCHEMBL2011167 0.81 RAB9A (0.79) SMN1; SMN2RAB9AKDM4EGAANPC1
SCHEMBL289554 0.81 SMN1; SMN2 (0.85) SMN1; SMN2RAB9AKDM4EGAANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5614520-A 2-arylthiazole derivatives and pharmaceutical composition thereof TEIJIN LIMITED (JP) 1997-03-25 US disclosed
EP-0513379-B1 2-ARYLTHIAZOLE DERIVATIVE AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME TEIJIN LTD (JP) 1996-09-11 EP disclosed
EP-0513379-A1 2-ARYLTHIAZOLE DERIVATIVE AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME TEIJIN LIMITED (JP) 1992-11-19 EP disclosed