SCHEMBL8867673

SCHEMBL8867673

CCOC(=O)c1sc(-c2ccc(C(=O)c3ccccc3)cc2)nc1C

nearest known ligand 0.81

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 6/20 0.67
DBF4 Q9UBU7 6/20 0.67
TRPM8 Q7Z2W7 5/20 0.63
LMNA P02545 1/20 0.62
RARA P10276 1/20 0.58
RARB P10826 1/20 0.58
RARG P13631 1/20 0.58
ALDH1A1 P00352 2/20 0.57
KDM4E B2RXH2 1/20 0.57
SMN1; SMN2 Q16637 2/20 0.55
MAPT P10636 3/20 0.54
NPC1 O15118 2/20 0.54
HPGD P15428 2/20 0.54
RAB9A P51151 1/20 0.54
GAA P10253 1/20 0.52
CSNK1D P48730 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL289229 0.90 CDC7 (0.73) CDC7DBF4TRPM8LMNARARA
SCHEMBL1316281 0.90 CDC7 (0.77) CDC7DBF4TRPM8LMNARARA
SCHEMBL8867028 0.88 CDC7 (0.71) CDC7DBF4TRPM8LMNARARA
SCHEMBL2880861 0.85 CDC7 (0.67) CDC7DBF4TRPM8LMNARARA
SCHEMBL8867115 0.84 SMN1; SMN2 (0.77) LMNARARARARBRARGALDH1A1
SCHEMBL892889 0.84 CDC7 (0.77) CDC7DBF4TRPM8LMNAALDH1A1
SCHEMBL290013 0.84 CDC7 (0.68) CDC7DBF4TRPM8LMNARARA
SCHEMBL290384 0.83 CDC7 (0.75) CDC7DBF4TRPM8LMNAALDH1A1
SCHEMBL257340 0.82 NPC1 (0.59) CDC7DBF4TRPM8LMNAALDH1A1
SCHEMBL2885887 0.82 TRPM8 (0.78) CDC7DBF4TRPM8LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5614520-A 2-arylthiazole derivatives and pharmaceutical composition thereof TEIJIN LIMITED (JP) 1997-03-25 US disclosed
EP-0513379-B1 2-ARYLTHIAZOLE DERIVATIVE AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME TEIJIN LTD (JP) 1996-09-11 EP disclosed
EP-0513379-A1 2-ARYLTHIAZOLE DERIVATIVE AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME TEIJIN LIMITED (JP) 1992-11-19 EP disclosed