SCHEMBL8867321

SCHEMBL8867321

O=c1c(Cc2ccccc2)cn2c3c(cccc13)COc1ccccc1-2

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.37
HSD17B3 P37058 1/20 0.37
TSHR P16473 2/20 0.34
TP53 P04637 1/20 0.34
POLB P06746 1/20 0.34
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
XIAP P98170 2/20 0.33
TOP2A P11388 1/20 0.33
TOP2B Q02880 1/20 0.33
ALDH1A1 P00352 1/20 0.33
RIPK1 Q13546 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ALOX12 P18054 1/20 0.32
PIK3CG P48736 1/20 0.32
FEN1 P39748 1/20 0.32
NR1H2 P55055 1/20 0.32
CTRC Q99895 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8868135 0.84 TOP2A (0.38) HSD17B3TSHRTOP2ATOP2BALDH1A1
SCHEMBL30144051 0.61 POLB (0.51) THRBHSD17B3TSHRPOLBALDH1A1
SCHEMBL27691202 0.61 AKR1A1 (0.48) TSHRTP53ALDH1A1
SCHEMBL19971597 0.60 TOP2A (0.48) TOP2ATOP2B
SCHEMBL6807700 0.59 MEN1 (0.50) HSD17B3TSHRTP53POLBALDH1A1
Diphenylmethane SCHEMBL1064958 0.59 MAOA (0.74) ALDH1A1L3MBTL1
SCHEMBL11494803 0.58 PDE3B (0.43) ALDH1A1NR1H2CTRC
SCHEMBL17933754 0.58 HSD17B3 (0.51) HSD17B3TSHRALDH1A1L3MBTL1
SCHEMBL6836937 0.57 MAOA (0.34) ALDH1A1
SCHEMBL2398512 0.57 CYP11B1 (0.77)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5677296-A ANALGESICS, ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1997-10-14 US disclosed
US-5488046-A ANALGESICS G. D. SEARLE & CO. (US) 1996-01-30 US disclosed