SCHEMBL8869706

SCHEMBL8869706

CN(C)Cc1c[nH]c2ccc(Oc3cccc(C(F)(F)F)c3)cc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPM8 Q7Z2W7 2/20 0.47
CYP2D6 P10635 2/20 0.47
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 1/20 0.47
ALDH1A1 P00352 1/20 0.47
CYP3A4 P08684 1/20 0.47
TSHR P16473 1/20 0.47
CYP2C19 P33261 1/20 0.47
KMT2A Q03164 1/20 0.47
HSD17B10 Q99714 1/20 0.47
HTR1D P28221 6/20 0.47
HTR1B P28222 4/20 0.47
HTR1A P08908 2/20 0.47
HTR2A P28223 2/20 0.45
HTR6 P50406 2/20 0.45
HTR3E A5X5Y0 1/20 0.45
HTR3B O95264 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
HTR2C P28335 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8870467 0.89 HTR1D (0.61) TRPM8CYP2D6KMT2AHTR1DHTR1B
Oxalic Acid SCHEMBL8868671 0.83 KMT2A (0.66) TRPM8CYP2D6KMT2AHTR1DHTR1B
SCHEMBL8868820 0.82 TRPM8 (0.71) TRPM8KDM4ETSHRHTR1DHTR1B
Hydrochloric Acid SCHEMBL8870348 0.81 TRPM8 (0.70) TRPM8KDM4EMEN1TSHRKMT2A
SCHEMBL8869614 0.81 CSNK2A1 (0.49) TRPM8HTR1DHTR1BHTR1ATRPV1
SCHEMBL8868679 0.80 TRPV1 (0.42) TRPM8KMT2AHTR1DHTR1BHTR1A
SCHEMBL1196580 0.79 HTR1D (0.53) TRPM8CYP2D6KDM4EMEN1ALDH1A1
SCHEMBL8870437 0.79 HTR1D (0.52) TRPM8CYP2D6KDM4EMEN1ALDH1A1
SCHEMBL8869870 0.79 HTR1A (0.63) TRPM8CYP2D6KDM4EMEN1ALDH1A1
SCHEMBL8869671 0.79 TRPM8 (0.49) TRPM8CYP2D6KDM4EMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5637593-A MIGRAINE; HYPOTENSIVE AGENTS SMITHKLINE BEECHAM PLC (GB) 1997-06-10 US disclosed