SCHEMBL8869876

SCHEMBL8869876

CN(C)C(=O)Sc1ccc2c(c1)C(=O)CCC2

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.42
ALDH1A1 P00352 2/20 0.42
MAOA P21397 6/20 0.40
MAOB P27338 6/20 0.40
CYP2A6 P11509 1/20 0.40
BAZ2B Q9UIF8 1/20 0.40
PRKCI P41743 1/20 0.40
PBRM1 Q86U86 1/20 0.38
MEN1 O00255 1/20 0.36
MAPK1 P28482 1/20 0.36
KMT2A Q03164 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HSD17B1 P14061 1/20 0.36
GRM5 P41594 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7976822 0.77 ALDH1A1 (0.39) ACHEALDH1A1MAOAMAOBBAZ2B
SCHEMBL29649260 0.77 MAOA (0.48) MAOAMAOBCYP2A6BAZ2BPRKCI
SCHEMBL6076319 0.77 MAOA (0.48) MAOAMAOBCYP2A6BAZ2BPRKCI
SCHEMBL7714618 0.73 TYMS (0.45) MAOAMAOBCYP2A6BAZ2BPRKCI
SCHEMBL7237468 0.70 MAOA (0.48) ACHEALDH1A1MAOAMAOBCYP2A6
SCHEMBL315282 0.70 MAOA (0.53) MAOAMAOBCYP2A6BAZ2BPRKCI
SCHEMBL20244667 0.70 ALDH1A1 (0.53) ACHEALDH1A1KMT2ANPSR1
SCHEMBL18159338 0.69 NPC1 (0.53) ALDH1A1MAOAMAOBCYP2A6BAZ2B
SCHEMBL4455438 0.69 ALDH1A1 (0.54) ACHEALDH1A1CYP2A6
SCHEMBL30772981 0.69 ALDH1A1 (0.54) ACHEALDH1A1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607928-A Carbapenem derivatives containing a bicyclic ketone substituent and their use as anti-infectives ZENECA LIMITED (GB) 1997-03-04 US disclosed
EP-0695753-A1 Carbapenem derivatives containing a bicyclic substituent, process for their preparation, and their use ZENECA LIMITED (GB) 1996-02-07 EP disclosed