SCHEMBL8871049

SCHEMBL8871049

CCOC(=O)CNC(=O)n1ccnc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.42
LMNA P02545 2/20 0.42
PPID Q08752 2/20 0.42
GAA P10253 3/20 0.41
HSD17B10 Q99714 2/20 0.41
HPGD P15428 1/20 0.41
CYP17A1 P05093 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP21A2 P08686 1/20 0.41
CYP11B1 P15538 1/20 0.41
TBXAS1 P24557 3/20 0.40
KDM4E B2RXH2 2/20 0.39
TSHR P16473 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
MAPT P10636 2/20 0.39
MEN1 O00255 1/20 0.39
MITF O75030 1/20 0.39
KMT2A Q03164 1/20 0.39
ABL1 P00519 1/20 0.38
RIN1 Q13671 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18631522 0.82 L3MBTL1 (0.38) CYP17A1MAPT
SCHEMBL17285650 0.79 ALDH1A1 (0.35) ALDH1A1LMNACYP3A4TBXAS1SMN1; SMN2
SCHEMBL6808774 0.79 KMT2A (0.41) ALDH1A1MAPTKMT2AHTT
SCHEMBL21039172 0.77 ALDH1A1 (0.36) ALDH1A1TBXAS1SMN1; SMN2MAPT
SCHEMBL8872429 0.77 ALDH1A1 (0.44) ALDH1A1TBXAS1MAPT
SCHEMBL217356 0.77 ALDH1A1 (0.42) ALDH1A1LMNATBXAS1KDM4ETSHR
SCHEMBL5257422 0.76 QPCT (0.45) ALDH1A1LMNAGAASMN1; SMN2MEN1
SCHEMBL17517848 0.75 TBXAS1 (0.48) ALDH1A1GAATBXAS1KDM4ETSHR
SCHEMBL10407622 0.75 TBXAS1 (0.45) ALDH1A1LMNAGAATBXAS1KDM4E
SCHEMBL12150031 0.75 CYP26A1 (0.40) ALDH1A1TBXAS1KDM4ESMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5610144-A CHOLECYSTOKININ OR GASTRIN ANTAGONISTS; NERVOUS SYSTEM AND GASTROINTESTINAL DISORDERS RHONE-POULENC RORER S.A. (FR) 1997-03-11 US disclosed