SCHEMBL8873261

SCHEMBL8873261

CC=CCC1Cc2ccccc2C1=O

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
METAP1 P53582 4/20 0.58
ACHE P22303 7/20 0.52
CYP19A1 P11511 1/20 0.50
HTR2C P28335 2/20 0.45
HTR1A P08908 1/20 0.45
DRD2 P14416 1/20 0.45
HTR2A P28223 1/20 0.45
HTR7 P34969 1/20 0.45
HRH1 P35367 1/20 0.45
DRD3 P35462 1/20 0.45
HTR2B P41595 1/20 0.45
SIGMAR1 Q99720 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8873256 1.00 METAP1 (0.58) METAP1ACHECYP19A1HTR2CHTR1A
SCHEMBL8873267 1.00 METAP1 (0.58) METAP1ACHECYP19A1HTR2CHTR1A
SCHEMBL8596739 0.82 TYRO3 (0.40) METAP1ACHECYP19A1
SCHEMBL8596737 0.82 TYRO3 (0.40) METAP1ACHECYP19A1
SCHEMBL8874229 0.82 TYRO3 (0.40) METAP1ACHECYP19A1
SCHEMBL8364658 0.81 METAP1 (0.61) METAP1ACHECYP19A1HTR2CHTR1A
SCHEMBL28949987 0.81 METAP1 (0.51) METAP1ACHECYP19A1HTR2CHTR1A
SCHEMBL8595392 0.80 METAP1 (0.59) METAP1ACHEHTR2CHTR2AHTR2B
SCHEMBL8873299 0.80 METAP1 (0.59) METAP1ACHEHTR2CHTR2AHTR2B
SCHEMBL8595390 0.80 METAP1 (0.59) METAP1ACHEHTR2CHTR2AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5646173-A ANTISEROTONINE AGENTS; CENTRAL NERVOUS SYSTEM DISORDERS; ANTIDEPRESSANTS HOFFMANN-LA ROCHE INC. (US) 1997-07-08 US disclosed
EP-0657426-A2 Tricyclic pyrrole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1995-06-14 EP disclosed