SCHEMBL8874246

SCHEMBL8874246

O=c1[nH]c2ccccc2cc1CN1CC=C(CCc2ccccc2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.45
PARP1 P09874 3/20 0.42
IL4I1 Q96RQ9 4/20 0.41
DRD2 P14416 2/20 0.41
DRD4 P21917 2/20 0.41
DRD3 P35462 2/20 0.41
KDM4E B2RXH2 5/20 0.40
ALDH1A1 P00352 4/20 0.40
HRH4 Q9H3N8 1/20 0.40
MAPK1 P28482 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HPGD P15428 1/20 0.39
MAPT P10636 1/20 0.38
TSHR P16473 1/20 0.38
NPC1 O15118 1/20 0.38
HTT P42858 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CYP1A2 P05177 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8873570 0.90 KDR (0.45) KDRPARP1IL4I1DRD2DRD4
SCHEMBL9396362 0.84 HRH4 (0.51) DRD2DRD4DRD3HRH4
SCHEMBL8875223 0.82 PARP1 (0.58) PARP1DRD2DRD4DRD3KDM4E
SCHEMBL9392973 0.78 HRH4 (0.49) DRD2DRD4DRD3HRH4
SCHEMBL8874059 0.77 DRD2 (0.49) KDRPARP1IL4I1DRD2DRD4
SCHEMBL8875278 0.77 DRD2 (0.49) KDRPARP1IL4I1DRD2DRD4
Oxalic Acid SCHEMBL8683797 0.76 HRH4 (0.45) DRD2DRD4DRD3HRH4NPSR1
SCHEMBL8984029 0.75 SIGMAR1 (0.50) DRD2DRD4DRD3HTT
SCHEMBL9091956 0.75 BCHE (0.57) DRD2DRD4DRD3KDM4EALDH1A1
SCHEMBL1813854 0.74 KDR (0.60) KDRPARP1DRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607946-A Quinolone derivatives as dopamine D4 ligands MERCK SHARP & DOHME LTD. (GB) 1997-03-04 US disclosed