SCHEMBL8875223

SCHEMBL8875223

O=c1[nH]c2ccccc2cc1CN1CC=C(c2ccccc2)CC1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.58
DRD4 P21917 4/20 0.56
KDM4E B2RXH2 6/20 0.53
MAPT P10636 6/20 0.53
GAA P10253 4/20 0.50
HTT P42858 1/20 0.50
CASP1 P29466 1/20 0.50
HBB P68871 1/20 0.50
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
ATM Q13315 1/20 0.49
DRD2 P14416 2/20 0.49
ALDH1A1 P00352 2/20 0.47
CYP3A4 P08684 1/20 0.47
ALOX15 P16050 1/20 0.47
TSHR P16473 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
DRD3 P35462 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8873570 0.83 KDR (0.45) PARP1DRD4KDM4EDRD2ALDH1A1
SCHEMBL8683088 0.83 DRD4 (0.60) PARP1DRD4KDM4EMAPTGAA
SCHEMBL8068175 0.82 PARP1 (0.66) PARP1DRD4KDM4EMAPTGAA
SCHEMBL8874246 0.82 KDR (0.45) PARP1DRD4KDM4EMAPTHTT
SCHEMBL8874059 0.81 DRD2 (0.49) PARP1DRD4KDM4EKMT2ADRD2
SCHEMBL8875278 0.81 DRD2 (0.49) PARP1DRD4KDM4EKMT2ADRD2
SCHEMBL1813854 0.80 KDR (0.60) PARP1DRD4HTTDRD2DRD3
SCHEMBL3395249 0.78 DRD4 (0.71) PARP1DRD4KDM4EMAPTGAA
SCHEMBL8874381 0.77 KDM4E (0.52) DRD4KDM4EMAPTGAAHTT
SCHEMBL8875085 0.75 DRD4 (0.53) PARP1DRD4KDM4EMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607946-A Quinolone derivatives as dopamine D4 ligands MERCK SHARP & DOHME LTD. (GB) 1997-03-04 US disclosed