SCHEMBL8875138

SCHEMBL8875138

COc1ccccc1C1(O)CCC(=O)C2CNCC21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.46
CHRM2 P08172 1/20 0.41
CHRM4 P08173 1/20 0.41
CHRM5 P08912 1/20 0.41
CHRM1 P11229 1/20 0.41
CHRM3 P20309 1/20 0.41
KMT2A Q03164 2/20 0.41
TACR1 P25103 3/20 0.40
CYP3A4 P08684 2/20 0.37
MAPT P10636 2/20 0.37
MEN1 O00255 1/20 0.37
TSHR P16473 1/20 0.37
CYP2C19 P33261 1/20 0.37
ALDH1A1 P00352 1/20 0.36
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35
OPRL1 P41146 1/20 0.35
SCN9A Q15858 1/20 0.34
TP53 P04637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8874853 0.99 SIGMAR1 (0.45) SIGMAR1CHRM2CHRM4CHRM5CHRM1
Hydrochloric Acid SCHEMBL8874914 0.76 SIGMAR1 (0.49) SIGMAR1CHRM2CHRM4CHRM5CHRM1
SCHEMBL8544913 0.75 TACR1 (0.56) SIGMAR1CHRM2CHRM4CHRM5CHRM1
SCHEMBL8873371 0.75 SIGMAR1 (0.48) SIGMAR1CHRM2CHRM4CHRM5CHRM1
SCHEMBL8875253 0.74 CHRM4 (0.44) SIGMAR1CHRM2CHRM4CHRM5CHRM1
Hydrochloric Acid SCHEMBL9241561 0.74 TACR1 (0.55) SIGMAR1CHRM2CHRM4CHRM5CHRM1
Hydrochloric Acid SCHEMBL8956731 0.74 TACR1 (0.55) SIGMAR1CHRM2CHRM4CHRM5CHRM1
Hydrochloric Acid SCHEMBL7886015 0.74 TACR1 (0.55) SIGMAR1CHRM2CHRM4CHRM5CHRM1
SCHEMBL8874681 0.73 SIGMAR1 (0.46) SIGMAR1CHRM2CHRM4CHRM5CHRM1
SCHEMBL8874475 0.72 TACR1 (0.57) SIGMAR1KMT2ATACR1CYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5624950-A USEFUL IN TREATMENT OF ANALGESIA, INFLAMMATION, ASTHMA, ALLERGIES, CENTRAL NERVOUS SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS, IMMUNE SYSTEM DISORDERS, ANTISPASMODIC AGENTS, ANTIEMETIC AGENTS RHONE-POULENC RORER S.A. (FR) 1997-04-29 US disclosed