SCHEMBL8874381

SCHEMBL8874381

O=c1[nH]c2ccccc2cc1CN1CCc2ccccc2C1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.52
KMT2A Q03164 2/20 0.52
GAA P10253 2/20 0.52
MAPT P10636 1/20 0.52
HTT P42858 1/20 0.52
TAAR1 Q96RJ0 1/20 0.52
ALDH1A1 P00352 4/20 0.52
HSD17B10 Q99714 1/20 0.52
DRD2 P14416 2/20 0.50
DRD4 P21917 2/20 0.50
DRD3 P35462 2/20 0.50
SPR P35270 1/20 0.48
POLB P06746 1/20 0.48
KDR P35968 1/20 0.47
IL4I1 Q96RQ9 1/20 0.46
DAO P14920 1/20 0.46
PKM P14618 1/20 0.46
DHFR P00374 1/20 0.46
MEN1 O00255 1/20 0.45
TSHR P16473 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8681907 0.81 DRD2 (0.68) KDM4EKMT2AGAAMAPTHTT
SCHEMBL8077800 0.81 PARP1 (0.54) KDM4EKMT2AGAAMAPTHTT
SCHEMBL8875223 0.77 PARP1 (0.58) KDM4EKMT2AGAAMAPTHTT
SCHEMBL6345975 0.76 SIGMAR1 (0.54) KMT2AALDH1A1DRD2IL4I1MEN1
SCHEMBL8875085 0.75 DRD4 (0.53) KDM4EMAPTHTTALDH1A1DRD2
SCHEMBL8873570 0.74 KDR (0.45) KDM4EALDH1A1HSD17B10DRD2DRD4
SCHEMBL8874246 0.73 KDR (0.45) KDM4EMAPTHTTALDH1A1HSD17B10
SCHEMBL8875278 0.72 DRD2 (0.49) KDM4EKMT2AALDH1A1DRD2DRD4
SCHEMBL8874059 0.72 DRD2 (0.49) KDM4EKMT2AALDH1A1DRD2DRD4
SCHEMBL8874997 0.72 DRD4 (0.57) KDM4EKMT2AGAAMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607946-A Quinolone derivatives as dopamine D4 ligands MERCK SHARP & DOHME LTD. (GB) 1997-03-04 US disclosed