SCHEMBL8875008

SCHEMBL8875008

Cc1cc(CCCOc2ccc(C(=N)NO)cc2C)on1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ALDH1A1 P00352 2/20 0.38
HDAC6 Q9UBN7 1/20 0.36
KDM4E B2RXH2 1/20 0.36
TP53 P04637 1/20 0.36
ALOX15 P16050 1/20 0.36
IGF1R P08069 2/20 0.34
FGFR1 P11362 2/20 0.34
KDR P35968 2/20 0.34
THRA P10827 1/20 0.33
THRB P10828 1/20 0.33
INSR P06213 1/20 0.33
F2 P00734 1/20 0.33
PLAU P00749 1/20 0.33
ST14 Q9Y5Y6 1/20 0.33
USP2 O75604 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8136108 0.86 NR1I2 (0.45) NR1I2CYP3A4CYP2D6THRATHRB
SCHEMBL8138666 0.85 NR1I2 (0.54) NR1I2CYP3A4CYP2D6MEN1KMT2A
SCHEMBL8876220 0.85 HDAC6 (0.46) NR1I2CYP3A4CYP2D6MEN1KMT2A
SCHEMBL8136126 0.84 PRSS1 (0.49) MEN1KMT2AALDH1A1KDM4ETHRA
SCHEMBL8874123 0.80 NR1I2 (0.47) NR1I2CYP3A4CYP2D6MEN1KMT2A
SCHEMBL9176420 0.80 NR1I2 (0.49) NR1I2CYP3A4CYP2D6MEN1KMT2A
SCHEMBL8130660 0.80 CYP3A4 (0.43) NR1I2CYP3A4CYP2D6MEN1KMT2A
SCHEMBL8875258 0.78 NR1I2 (0.44) NR1I2CYP3A4CYP2D6MEN1KMT2A
SCHEMBL8875413 0.78 NR1I2 (0.47) NR1I2CYP3A4CYP2D6MEN1KMT2A
SCHEMBL25801629 0.78 THRA (0.48) MEN1KMT2AKDM4ETP53ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5643929-A TREATMENT OF PICORNAVIRAL OR RHINOVIRUS AND CHEMICAL INTERMEDIATES SANOFI WINTHROP, INC. (US) 1997-07-01 US disclosed
US-5464848-A 1,2,4-oxadiazolyl-phenoxyalkylisoxazoles and their use as antiviral agents STERLING WINTHROP INC. (US) 1995-11-07 US disclosed