SCHEMBL8876808

SCHEMBL8876808

CC(C)c1nc(-c2cccc3ccccc23)cc(-c2ccc(F)cc2)c1C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
PPARG P37231 4/20 0.44
PPARA Q07869 4/20 0.44
FABP3 P05413 1/20 0.43
FABP4 P15090 1/20 0.43
FABP5 Q01469 1/20 0.43
DHODH Q02127 2/20 0.43
DHFR P00374 1/20 0.43
ALKBH5 Q6P6C2 1/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
AKR1C3 P42330 1/20 0.42
AKR1C2 P52895 1/20 0.42
GRM2 Q14416 1/20 0.41
HMGCR P04035 1/20 0.41
MCL1 Q07820 1/20 0.41
ACMSD Q8TDX5 1/20 0.41
GPR84 Q9NQS5 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8878154 0.86 DHODH (0.44) FABP3FABP4FABP5DHODHDHFR
SCHEMBL8879993 0.86 HMGCR (0.49) FABP3FABP4FABP5DHODHKDM4E
SCHEMBL8877432 0.81 HMGCR (0.44) PPARGPPARAGRM2HMGCR
SCHEMBL8877852 0.81 GCGR (0.49) HMGCR
SCHEMBL8877871 0.81 PTGDR2 (0.42) MEN1KMT2ADHODHDHFRALKBH5
SCHEMBL8876825 0.80 PPARA (0.46) MEN1KMT2APPARAFABP3FABP4
SCHEMBL8878856 0.80 GCGR (0.46) FABP3FABP4FABP5HMGCR
SCHEMBL8878198 0.79 DHODH (0.40) DHODHHMGCR
SCHEMBL8876862 0.79 HMGCR (0.42) PPARGPPARAHMGCR
SCHEMBL8880943 0.78 GCGR (0.45) PPARAFABP3FABP4FABP5DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691322-A Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1997-11-25 US disclosed
US-5686433-A CHOLESTEROL BIOSYNTHESIS INHIBITION E.R. SQUIBB & SONS, INC. (US) 1997-11-11 US disclosed
US-5506219-A ANTICHOLESTEROL AND ANTILIPEMIC AGENTS E. R. SQUIBB & SONS, INC. (US) 1996-04-09 US disclosed