SCHEMBL8877112

SCHEMBL8877112

COc1ccccc1N1CCN(CCNCc2cccc3c(=O)c(C)c(-c4ccccc4)oc23)CC1

nearest known ligand 0.72

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 7/20 0.68
ADRA1A P35348 6/20 0.68
ADRA1D P25100 5/20 0.68
ADRA1B P35368 5/20 0.68
ALDH1A1 P00352 1/20 0.61
LMNA P02545 1/20 0.61
CD274 Q9NZQ7 1/20 0.54
HTR2A P28223 2/20 0.49
HTR7 P34969 2/20 0.49
HTR6 P50406 1/20 0.49
DRD2 P14416 3/20 0.47
DRD3 P35462 3/20 0.47
DRD4 P21917 2/20 0.47
ADRA2A P08913 1/20 0.47
DRD1 P21728 1/20 0.47
DRD5 P21918 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8876154 0.95 ADRA1A (0.73) HTR1AADRA1AADRA1DADRA1BALDH1A1
Hydrochloric Acid SCHEMBL8876536 0.94 ADRA1A (0.72) HTR1AADRA1AADRA1DADRA1BALDH1A1
SCHEMBL8876730 0.89 HTR1A (0.64) HTR1AADRA1AADRA1DADRA1BALDH1A1
SCHEMBL8877818 0.86 HTR1A (0.69) HTR1AADRA1AADRA1DADRA1BALDH1A1
SCHEMBL8876383 0.86 HTR1A (0.69) HTR1AADRA1AADRA1DADRA1BALDH1A1
SCHEMBL8875919 0.86 HTR1A (0.78) HTR1AADRA1AADRA1DADRA1BALDH1A1
Hydrochloric Acid SCHEMBL8875648 0.86 HTR1A (0.69) HTR1AADRA1AADRA1DADRA1BALDH1A1
SCHEMBL8874490 0.86 HTR1A (0.66) HTR1AADRA1AADRA1DADRA1BALDH1A1
SCHEMBL8875779 0.86 HTR1A (0.69) HTR1AADRA1AADRA1DADRA1BALDH1A1
SCHEMBL8876843 0.85 HTR1A (0.66) HTR1AADRA1AADRA1DADRA1BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5605896-A Bicyclic heterocyclic derivatives having α1 adrenergic and 5HT1A activities RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1997-02-25 US disclosed
US-5403842-A Adrenergic blocking and antiserotonine agents; urogenital disorders including spasms of the urethral tract and prostrate problems RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1995-04-04 US disclosed
EP-0558245-A1 Heterobicyclic compounds as antagogists of alpha-1 adrenergic and SHT1A receptors RECORDATI S.A. CHEMICAL and PHARMACEUTICAL COMPANY (CH) 1993-09-01 EP disclosed