SCHEMBL8877779

SCHEMBL8877779

C[C@H](N)C(=O)N(CCC(C)(C)c1ccc2ccccc2c1)C(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 2/20 0.38
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
KCNH2 Q12809 1/20 0.34
CPB2 Q96IY4 1/20 0.34
CTSB P07858 1/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
GABRB1 P18505 1/20 0.32
GABRB2 P47870 1/20 0.32
GRIN2D O15399 1/20 0.32
GRIN3B O60391 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2A Q12879 1/20 0.32
GRIN2B Q13224 1/20 0.32
GRIN2C Q14957 1/20 0.32
GRIN3A Q8TCU5 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8771876 0.75 KDM4E (0.41) PPARAKDM4EALDH1A1
SCHEMBL8771976 0.71 FDPS (0.38) CYP3A4CYP2D6SLC6A4ALDH1A1
SCHEMBL10627360 0.69 L3MBTL1 (0.32) CYP3A4CYP2D6SLC6A4KCNH2CPB2
SCHEMBL6832915 0.66 SMN1; SMN2 (0.40) CTSBCTSSCTSKGABRB1GABRB2
SCHEMBL12805323 0.66 CTSB (0.48) CTSBCTSSCTSK
SCHEMBL7344398 0.66 GRIK1 (0.36) CPB2CTSK
SCHEMBL7346071 0.66 GRIK1 (0.36) CPB2CTSK
SCHEMBL6295389 0.66 HDAC6 (0.32)
SCHEMBL28195146 0.66 MEN1 (0.33) GABRB1GABRB2
SCHEMBL28195145 0.66 MEN1 (0.33) GABRB1GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5668128-A INHIBITORS OF THIOL PROTEASE, PROPHYLAXIS AND TREATMENT OF BONE DISEASES, OSTEOPOROSIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-09-16 US disclosed