SCHEMBL8877862

SCHEMBL8877862

Cc1cc(F)ccc1-c1cc(-c2ccccc2)nc(C(C)C)c1C=O

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 4/20 0.44
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
DHODH Q02127 1/20 0.35
AR P10275 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9849071 0.88 HMGCR (0.37) HMGCRKDM4EALDH1A1GLAGAA
SCHEMBL8875477 0.85 HMGCR (0.42) HMGCRDHODH
SCHEMBL8878341 0.85 HMGCR (0.57) HMGCR
SCHEMBL8877954 0.81 DHODH (0.43) HMGCRDHODH
SCHEMBL8877555 0.79 HMGCR (0.48) HMGCR
SCHEMBL8878729 0.79 SQOR (0.39) HMGCRKDM4EALDH1A1L3MBTL1
SCHEMBL8878236 0.78 HMGCR (0.43) HMGCR
SCHEMBL8952918 0.78 HMGCR (0.43) HMGCR
SCHEMBL8876796 0.77 HMGCR (0.46) HMGCR
SCHEMBL8953141 0.76

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691322-A Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1997-11-25 US disclosed
US-5686433-A CHOLESTEROL BIOSYNTHESIS INHIBITION E.R. SQUIBB & SONS, INC. (US) 1997-11-11 US disclosed
US-5506219-A ANTICHOLESTEROL AND ANTILIPEMIC AGENTS E. R. SQUIBB & SONS, INC. (US) 1996-04-09 US disclosed