SCHEMBL8877873

SCHEMBL8877873

CC(C)c1nc(C2CCCCC2)cc(-c2ccc(F)cc2)c1C=O

nearest known ligand 0.62

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 7/20 0.62
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40
APP P05067 1/20 0.38
GCGR P47871 2/20 0.37
MAPK14 Q16539 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9849223 0.88 HMGCR (0.53) HMGCRADORA2AADORA1GCGRMAPK14
SCHEMBL8876720 0.85 HMGCR (0.59) HMGCRADORA2AADORA1APPGCGR
SCHEMBL8879043 0.81 HMGCR (0.54) HMGCRADORA2AADORA1APPGCGR
SCHEMBL8878207 0.80 HMGCR (0.55) HMGCRADORA2AADORA1GCGR
SCHEMBL8949911 0.80 HMGCR (0.53) HMGCRADORA2AADORA1APPGCGR
SCHEMBL8878341 0.79 HMGCR (0.57) HMGCRADORA2AADORA1
SCHEMBL8878262 0.79 HMGCR (0.52) HMGCRADORA2AADORA1GCGR
SCHEMBL9022533 0.77 HMGCR (1.00) HMGCR
SCHEMBL6961433 0.77 HMGCR (0.54) HMGCRGCGR
SCHEMBL8877661 0.77 GCGR (0.46) HMGCRGCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691322-A Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1997-11-25 US disclosed
US-5686433-A CHOLESTEROL BIOSYNTHESIS INHIBITION E.R. SQUIBB & SONS, INC. (US) 1997-11-11 US disclosed
US-5506219-A ANTICHOLESTEROL AND ANTILIPEMIC AGENTS E. R. SQUIBB & SONS, INC. (US) 1996-04-09 US disclosed