SCHEMBL9849223

SCHEMBL9849223

CC(CI)c1nc(C2CCCCC2)cc(-c2ccc(F)cc2)c1C=O

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 6/20 0.53
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37
GCGR P47871 1/20 0.36
MAPK14 Q16539 1/20 0.36
KDM4E B2RXH2 2/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
HTT P42858 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34
GRM2 Q14416 1/20 0.34
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8877873 0.88 HMGCR (0.62) HMGCRADORA2AADORA1GCGRMAPK14
SCHEMBL9849239 0.82 HMGCR (0.48) HMGCRADORA2AADORA1GCGRMAPK14
SCHEMBL9849206 0.77 MEN1 (0.42) HMGCRADORA2AMAPK14KDM4ELMNA
SCHEMBL8876720 0.74 HMGCR (0.59) HMGCRADORA2AADORA1GCGR
SCHEMBL8878207 0.73 HMGCR (0.55) HMGCRADORA2AADORA1GCGR
SCHEMBL8949911 0.73 HMGCR (0.53) HMGCRADORA2AADORA1GCGRMAPK14
SCHEMBL8879043 0.72 HMGCR (0.54) HMGCRADORA2AADORA1GCGRKDM4E
SCHEMBL9022533 0.69 HMGCR (1.00) HMGCR
SCHEMBL9849071 0.69 HMGCR (0.37) HMGCRKDM4EL3MBTL1
SCHEMBL8878262 0.68 HMGCR (0.52) HMGCRADORA2AADORA1GCGRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0444533-A2 Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1991-09-04 EP disclosed