SCHEMBL8877993

SCHEMBL8877993

Cc1c(CCCC(=O)O)c2cc(Cl)ccc2n1Cc1ccc(Cl)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 9/20 0.63
MEN1 O00255 1/20 0.60
RGS12 O14924 1/20 0.60
ALDH1A1 P00352 1/20 0.60
LMNA P02545 1/20 0.60
CYP1A2 P05177 1/20 0.60
CYP3A4 P08684 1/20 0.60
MAPT P10636 1/20 0.60
CYP2C9 P11712 1/20 0.60
PKM P14618 1/20 0.60
TSHR P16473 1/20 0.60
NFKB1 P19838 1/20 0.60
MAPK1 P28482 1/20 0.60
CYP2C19 P33261 1/20 0.60
GNAI1 P63096 1/20 0.60
PMP22 Q01453 1/20 0.60
KMT2A Q03164 1/20 0.60
HIF1A Q16665 1/20 0.60
PTGES O14684 1/20 0.57
ALOX5 P09917 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8878924 0.93 PLA2G2A (0.59) PLA2G2AMEN1RGS12ALDH1A1LMNA
SCHEMBL8876342 0.93 PLA2G2A (0.59) PLA2G2AMEN1RGS12ALDH1A1LMNA
SCHEMBL8876716 0.91 PLA2G2A (0.59) PLA2G2AMEN1RGS12ALDH1A1LMNA
SCHEMBL3246296 0.87 PTGS2 (0.59) PLA2G2AMEN1RGS12ALDH1A1LMNA
SCHEMBL8877434 0.84 PLA2G2A (0.62) PLA2G2ATHRATHRBPTGS2
SCHEMBL8876622 0.82 PLA2G2A (0.60) PLA2G2ALMNAKMT2APTGESALOX5
SCHEMBL8876095 0.82 AKR1A1 (0.53) PLA2G2AMEN1RGS12ALDH1A1LMNA
SCHEMBL3001920 0.80 PLA2G2A (0.67) PLA2G2AMEN1RGS12ALDH1A1LMNA
SCHEMBL9741283 0.79 PTGES2 (0.57) MEN1RGS12ALDH1A1LMNACYP1A2
SCHEMBL7196880 0.79 PTGS2 (0.79) PLA2G2AMEN1RGS12ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996037467-A1 N-BENZYLINDOL-3-YL BUTANOIC ACID DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS MERCK FROSST CANADA INC. (CA) 1996-11-28 WO claimed
US-5639780-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS MERCK FROSST CANADA, INC. (CA) 1997-06-17 US disclosed