SCHEMBL8878013

SCHEMBL8878013

C#Cc1c(-c2ccc(F)cc2)cc(-c2ccccc2)nc1C(C)C

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SQOR Q9Y6N5 6/20 0.53
ADORA2A P29274 1/20 0.52
ADORA1 P30542 1/20 0.52
HMGCR P04035 2/20 0.45
TOP1 P11387 2/20 0.44
HPGD P15428 2/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
PTK2B Q14289 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9637289 0.85 SQOR (0.49) SQORADORA2AADORA1HMGCRHPGD
SCHEMBL8878729 0.85 SQOR (0.39) SQORADORA2AADORA1HMGCRHPGD
SCHEMBL8878416 0.83 SQOR (0.39) SQORADORA2AADORA1
SCHEMBL9635988 0.82 SQOR (0.48) SQORADORA2AADORA1HMGCRHPGD
SCHEMBL9636079 0.82 SQOR (0.48) SQORADORA2AADORA1HMGCRHPGD
SCHEMBL10024048 0.81 SQOR (0.48) SQORADORA2AADORA1HMGCRTOP1
SCHEMBL8877328 0.79 SQOR (0.53) SQORHMGCR
SCHEMBL8846077 0.79 HMGCR (0.54) SQORADORA2AADORA1HMGCRTOP1
SCHEMBL9636049 0.79 SQOR (0.51) SQORADORA2AADORA1HMGCRHPGD
SCHEMBL8877410 0.78 HMGCR (0.45) SQORADORA2AADORA1HMGCRTOP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691322-A Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1997-11-25 US disclosed
US-5686433-A CHOLESTEROL BIOSYNTHESIS INHIBITION E.R. SQUIBB & SONS, INC. (US) 1997-11-11 US disclosed
US-5506219-A ANTICHOLESTEROL AND ANTILIPEMIC AGENTS E. R. SQUIBB & SONS, INC. (US) 1996-04-09 US disclosed
EP-0356788-A2 Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1990-03-07 EP disclosed