SCHEMBL8846077

SCHEMBL8846077

[CH]=Cc1c(-c2ccc(F)cc2)cc(-c2ccccc2)nc1C(C)C

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 4/20 0.54
SQOR Q9Y6N5 1/20 0.44
TOP1 P11387 2/20 0.44
ADORA2A P29274 1/20 0.43
ADORA1 P30542 1/20 0.43
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
HPGD P15428 1/20 0.41
CYP2C19 P33261 1/20 0.41
PTK2B Q14289 1/20 0.41
GCGR P47871 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8225619 0.87 HMGCR (0.54) HMGCRSQORTOP1ADORA2AADORA1
SCHEMBL8878341 0.87 HMGCR (0.57) HMGCRSQORTOP1ADORA2AADORA1
SCHEMBL8878203 0.85 HMGCR (0.57) HMGCRSQORTOP1ADORA2AADORA1
SCHEMBL8878191 0.85 HMGCR (0.57) HMGCRSQORTOP1ADORA2AADORA1
SCHEMBL8876495 0.84 HMGCR (0.54) HMGCRSQORTOP1ADORA2AADORA1
SCHEMBL22604014 0.83 HMGCR (0.56) HMGCRSQOR
SCHEMBL8953098 0.83 HMGCR (0.58) HMGCR
SCHEMBL8953106 0.83 HMGCR (0.58) HMGCR
SCHEMBL10024048 0.81 SQOR (0.48) HMGCRSQORTOP1ADORA2AADORA1
SCHEMBL8878013 0.79 SQOR (0.53) HMGCRSQORTOP1ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0641762-B1 Process for preparation of 5-hydroxy-3-ketoester derivative and optically active substance thereof UBE INDUSTRIES (JP) 1997-05-28 EP disclosed
US-5457225-A Process for preparation of 5-hydroxy-3-ketoester derivative and optically active substance thereof UBE INDUSTRIES LTD. (JP) 1995-10-10 US disclosed
EP-0641762-A1 Process for preparation of 5-hydroxy-3-ketoester derivative and optically active substance thereof UBE INDUSTRIES, LTD. (JP) 1995-03-08 EP disclosed