SCHEMBL8878086

SCHEMBL8878086

COC(=O)CC(=O)c1cc(F)c(F)c(F)c1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
MAPK1 P28482 1/20 0.42
GAA P10253 2/20 0.40
SMN1; SMN2 Q16637 4/20 0.38
TDP1 Q9NUW8 1/20 0.38
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
MAPT P10636 3/20 0.35
CRBN Q96SW2 1/20 0.35
ATM Q13315 1/20 0.34
MGAM O43451 1/20 0.34
SI P14410 1/20 0.34
MGAM2 Q2M2H8 1/20 0.34
CES2 O00748 2/20 0.34
CES1 P23141 2/20 0.34
HSP90AB1 P08238 1/20 0.34
NPC1 O15118 2/20 0.33
HTT P42858 2/20 0.33
RAB9A P51151 2/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1185918 0.85 ALDH1A1 (0.44) ALDH1A1MAPK1GAASMN1; SMN2TDP1
SCHEMBL8877353 0.85 GAA (0.41) ALDH1A1MAPK1GAASMN1; SMN2MEN1
SCHEMBL30958584 0.85 ALDH1A1 (0.44) ALDH1A1MAPK1GAASMN1; SMN2TDP1
SCHEMBL7245515 0.83 SMN1; SMN2 (0.41) ALDH1A1MAPK1GAASMN1; SMN2TDP1
SCHEMBL8876484 0.81 GAA (0.42) ALDH1A1GAASMN1; SMN2MEN1KMT2A
Acetic Acid SCHEMBL8870017 0.81 ALDH1A1 (0.41) ALDH1A1MAPK1GAASMN1; SMN2TDP1
SCHEMBL1187294 0.79 PTPN1 (0.38) ALDH1A1MAPK1SMN1; SMN2TDP1CRBN
SCHEMBL30194898 0.79 PTPN1 (0.38) ALDH1A1MAPK1SMN1; SMN2TDP1CRBN
SCHEMBL1994444 0.79 MAPT (0.43) ALDH1A1GAASMN1; SMN2TDP1MAPT
SCHEMBL29162697 0.78 CES2 (0.48) ALDH1A1MAPK1GAASMN1; SMN2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5672708-A Process for the preparation of N-arylaminoacrylic acid derivatives and the use of N-arylaminoacrylic acid derivatives thus prepared for the preparation of 4-quinolone-3-carboxylic acid derivatives BAYER AKTIENGESELLSCHAFT (DE) 1997-09-30 US disclosed
EP-0239992-B1 PROCESS FOR THE PREPARATION OF 2,3,4,5-TETRAFLUOROBENZOYL ACETATES WARNER-LAMBERT COMPANY (US) 1989-09-06 EP disclosed
US-4772706-A Process for quinoline-3-carboxylic acid antibacterial agents WARNER-LAMBERT COMPANY (US) 1988-09-20 US disclosed
EP-0239992-A1 Process for the preparation of 2,3,4,5-tetrafluorobenzoyl acetates WARNER-LAMBERT COMPANY (US) 1987-10-07 EP disclosed
EP-0239992-A1 Process for the preparation of 2,3,4,5-tetrafluorobenzoyl acetates WARNER-LAMBERT COMPANY (US) 1987-10-07 EP disclosed
EP-0236673-A2 Process for quinoline-3-carboxylic acid antibacterial agents WARNER-LAMBERT COMPANY (US) 1987-09-16 EP disclosed
US-4689423-A Process for the preparation of 2,3,4,5-tetrafluorobenzoyl acetates WARNER-LAMBERT COMPANY (US) 1987-08-25 US disclosed
US-4689423-A Process for the preparation of 2,3,4,5-tetrafluorobenzoyl acetates WARNER-LAMBERT COMPANY (US) 1987-08-25 US disclosed