SCHEMBL8878166

SCHEMBL8878166

COc1ccccc1N1CCN(c2c(F)cc3c(=O)c(C(=O)OCCN4CCOCC4)cn(C)c3c2OC(F)F)CC1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
HTR4 Q13639 4/20 0.45
ADORA2B P29275 3/20 0.45
DRD2 P14416 4/20 0.40
DRD3 P35462 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
ADRA1A P35348 1/20 0.40
KDM4E B2RXH2 3/20 0.39
HPGD P15428 2/20 0.39
HSD17B10 Q99714 1/20 0.39
AKR1C3 P42330 1/20 0.39
DRD4 P21917 2/20 0.38
HRH2 P25021 1/20 0.38
HRH1 P35367 1/20 0.38
LMNA P02545 1/20 0.38
GLA P06280 1/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8878202 0.85 KDM4E (0.44) ALDH1A1SMN1; SMN2KDM4EHPGDHSD17B10
SCHEMBL8878155 0.79 KDM4E (0.47) ALDH1A1DRD3SMN1; SMN2KDM4EHPGD
SCHEMBL8732186 0.79 KDM4E (0.45) ALDH1A1HTR4KDM4EHPGDHSD17B10
SCHEMBL8735561 0.77 KDM4E (0.52) ALDH1A1DRD3SMN1; SMN2KDM4EHPGD
SCHEMBL8880183 0.75 KCNH2 (0.57) ALDH1A1KDM4EHPGDHSD17B10LMNA
Hydrochloric Acid SCHEMBL8732413 0.74 KCNH2 (0.56) ALDH1A1KDM4EHPGDHSD17B10LMNA
SCHEMBL8880495 0.72 HTR4 (0.40) ALDH1A1HTR4DRD3KDM4EHPGD
SCHEMBL8057309 0.71 KDM4E (0.46) ALDH1A1DRD2DRD3SMN1; SMN2KDM4E
SCHEMBL8877142 0.70 KDM4E (0.39) ALDH1A1HTR4SMN1; SMN2KDM4EHPGD
SCHEMBL24177747 0.70 ALDH1A1 (0.97) ALDH1A1SMN1; SMN2KDM4EHPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5519016-A Aryl group- or aromatic heterocyclic group-substituted aminoquinolone derivatives and anti-HIV agent UBE INDUSTRIES, LTD. (JP) 1996-05-21 US claimed
EP-0572259-A1 Aminoquinolone derivatives as anti-HIV agents UBE INDUSTRIES, LTD. (JP) 1993-12-01 EP claimed
US-5688791-A COMPOUNDS FOR TREATMENNT OF VIRAL DISEASES SUCH AS AIDS UBE INDUSTRIES, LTD. (JP) 1997-11-18 US disclosed
US-5519016-A Aryl group- or aromatic heterocyclic group-substituted aminoquinolone derivatives and anti-HIV agent UBE INDUSTRIES, LTD. (JP) 1996-05-21 US disclosed
EP-0572259-A1 Aminoquinolone derivatives as anti-HIV agents UBE INDUSTRIES, LTD. (JP) 1993-12-01 EP disclosed