SCHEMBL8878809

SCHEMBL8878809

Cc1c(CCC(C)C(=O)O)c2cc(Cl)ccc2n1Cc1ccc(Br)cc1F

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.48
AKR1A1 P14550 1/20 0.48
PTGS2 P35354 3/20 0.42
PLA2G2A P14555 1/20 0.42
MAPT P10636 3/20 0.41
PTGES O14684 1/20 0.41
ALOX5 P09917 1/20 0.41
MEN1 O00255 1/20 0.39
RGS12 O14924 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
PKM P14618 1/20 0.39
TSHR P16473 1/20 0.39
NFKB1 P19838 1/20 0.39
MAPK1 P28482 1/20 0.39
CYP2C19 P33261 1/20 0.39
GNAI1 P63096 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8876095 0.87 AKR1A1 (0.53) AKR1B1AKR1A1PTGS2PLA2G2AMAPT
SCHEMBL8878179 0.87 PTGS2 (0.54) PTGS2PLA2G2AMAPTPTGESALOX5
SCHEMBL8878139 0.75 PTGS2 (0.71) PTGS2PLA2G2AMAPTMEN1RGS12
SCHEMBL8878924 0.74 PLA2G2A (0.59) PTGS2PLA2G2AMAPTPTGESALOX5
SCHEMBL3246296 0.72 PTGS2 (0.59) PTGS2PLA2G2AMAPTPTGESALOX5
SCHEMBL8876716 0.72 PLA2G2A (0.59) PTGS2PLA2G2AMAPTPTGESALOX5
SCHEMBL8877140 0.71 PTGS2 (0.55) PTGS2PLA2G2AMAPTPTGESALOX5
SCHEMBL9056716 0.71 AKR1B1 (0.78) AKR1B1AKR1A1MEN1CYP1A2CYP2C9
SCHEMBL8877352 0.71 PTGS2 (0.53) PTGS2PLA2G2AMAPTPTGESALOX5
SCHEMBL10488007 0.71 AKR1B1 (0.85) AKR1B1AKR1A1MEN1CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996037467-A1 N-BENZYLINDOL-3-YL BUTANOIC ACID DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS MERCK FROSST CANADA INC. (CA) 1996-11-28 WO claimed
US-5639780-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS MERCK FROSST CANADA, INC. (CA) 1997-06-17 US disclosed
WO-1996037467-A1 N-BENZYLINDOL-3-YL BUTANOIC ACID DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS MERCK FROSST CANADA INC. (CA) 1996-11-28 WO disclosed