SCHEMBL8880508

SCHEMBL8880508

COC(=O)c1cccc(-c2ccc(Br)cc2)c1

nearest known ligand 0.64

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PLAU P00749 6/20 0.64
CA12 O43570 2/20 0.64
CA9 Q16790 2/20 0.64
CA1 P00915 1/20 0.64
CA2 P00918 1/20 0.64
ERN1 O75460 3/20 0.58
SLC6A3 Q01959 1/20 0.54
FNTA P49354 1/20 0.53
FNTB P49356 1/20 0.53
PGGT1B P53609 1/20 0.53
GABRG2 P18507 1/20 0.52
GABRB3 P28472 1/20 0.52
GABRA5 P31644 1/20 0.52
GABRA3 P34903 1/20 0.52
PLAT P00750 2/20 0.52
PLG P00747 1/20 0.52
EGFR P00533 1/20 0.51
CDK8 P49336 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27715902 0.89 CA12 (0.71) PLAUCA12CA9CA1CA2
SCHEMBL14898128 0.88 PLAU (0.59) PLAUCA12CA9CA1CA2
SCHEMBL68931 0.88 CA12 (0.69) PLAUCA12CA9CA1CA2
SCHEMBL67941 0.88 CA12 (0.68) PLAUCA12CA9CA1CA2
SCHEMBL29410906 0.86 TSHR (0.67) PLAUCA12CA9CA1CA2
SCHEMBL1221576 0.86 TSHR (0.67) PLAUCA12CA9CA1CA2
SCHEMBL1661764 0.85 CA12 (0.66) PLAUCA12CA9CA1CA2
SCHEMBL514 0.85 CA12 (0.66) PLAUCA12CA9CA1CA2
SCHEMBL30443216 0.85 CA12 (0.66) PLAUCA12CA9CA1CA2
SCHEMBL3359577 0.84 CA12 (0.65) PLAUCA12CA9CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed