SCHEMBL3359577

SCHEMBL3359577

COC(=O)c1cccc(-c2cccc(-c3ccccc3)c2)c1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.65
CA1 P00915 1/20 0.65
CA2 P00918 1/20 0.65
CA9 Q16790 1/20 0.65
TSHR P16473 1/20 0.64
GABRG2 P18507 1/20 0.64
GABRB3 P28472 1/20 0.64
GABRA5 P31644 1/20 0.64
GABRA3 P34903 1/20 0.64
KMO O15229 1/20 0.63
EGFR P00533 1/20 0.59
ERN1 O75460 1/20 0.59
PLAU P00749 3/20 0.58
RAB9A P51151 1/20 0.58
HDAC8 Q9BY41 1/20 0.58
NEK1 Q96PY6 1/20 0.57
AXL P30530 1/20 0.57
MAPT P10636 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
CDK8 P49336 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29410906 0.98 TSHR (0.67) CA12CA1CA2CA9TSHR
SCHEMBL1221576 0.98 TSHR (0.67) CA12CA1CA2CA9TSHR
Hydrochloric Acid SCHEMBL29506745 0.96 CA12 (0.65) CA12CA1CA2CA9TSHR
SCHEMBL27715902 0.94 CA12 (0.71) CA12CA1CA2CA9TSHR
SCHEMBL67941 0.92 CA12 (0.68) CA12CA1CA2CA9TSHR
SCHEMBL3032014 0.89 KMO (0.63) CA12CA1CA2CA9TSHR
SCHEMBL68931 0.89 CA12 (0.69) CA12CA1CA2CA9TSHR
SCHEMBL4257678 0.89 TSHR (0.63) CA12CA1CA2CA9TSHR
Trifluoroacetic Acid SCHEMBL27749215 0.89 PDK2 (0.57) CA12CA1CA2CA9TSHR
SCHEMBL27878777 0.88 TSHR (0.68) CA12CA1CA2CA9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7687482-B2 Bisphosphonate compounds and methods THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2010-03-30 US disclosed
EP-2001486-A2 BISPHOSPHONATE COMPOUNDS AND METHODS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2008-12-17 EP disclosed
US-20070275931-A1 BISPHOSPHONATE COMPOUNDS AND METHODS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2007-11-29 US disclosed
WO-2007109585-A2 BISPHOSPHONATE COMPOUNDS AND METHODS THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2007-09-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070275931-A1 BISPHOSPHONATE COMPOUNDS AND METHODS FDPS, GGPS1, FNTB CA12 2750/4885CA1 1681/4885CA2 679/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.