SCHEMBL8880685

SCHEMBL8880685

CN(C)C(=O)C(C)(C)C[O]

nearest known ligand 0.32

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.32
TSHR P16473 1/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
RIPK1 Q13546 2/20 0.31
MAPT P10636 1/20 0.31
NFKB1 P19838 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31
DRD4 P21917 1/20 0.31
OPRM1 P35372 1/20 0.31
DRD3 P35462 1/20 0.31
CYP3A4 P08684 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12293705 0.81 ALDH1A1 (0.30) ALDH1A1TSHRCYP3A4CYP2C9CYP2C19
SCHEMBL2740778 0.78 RIPK1 (0.47) RIPK1
SCHEMBL9607597 0.78 ALDH1A1 (0.32) ALDH1A1TSHRMEN1KMT2ARIPK1
SCHEMBL20857549 0.76 ALDH1A1 (0.30) ALDH1A1TSHR
SCHEMBL11809225 0.76 KDM4E (0.36) ALDH1A1TSHR
SCHEMBL5264333 0.76 ALDH1A1 (0.40) ALDH1A1TSHRMEN1KMT2ARIPK1
SCHEMBL11621506 0.76 ALDH1A1 (0.36) ALDH1A1TSHRDRD4OPRM1DRD3
SCHEMBL20221015 0.74 DRD4 (0.36) DRD4OPRM1DRD3
SCHEMBL24351044 0.72 DRD4 (0.32) DRD4OPRM1DRD3
SCHEMBL16841724 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5641778-A EXHIBIT RENIN-INHIBITING PROPERTIES AND CAN BE USED AS ANTIHYPERTENSIVE AGENTS CIBA-GEIGY CORPORATION (US) 1997-06-24 US disclosed
EP-0716077-A1 Aromatically substituted omega amino alcanoic acid amides and alcanoic diamides and their use as renine inhibitors CIBA-GEIGY AG (CH) 1996-06-12 EP disclosed