SCHEMBL8880802

SCHEMBL8880802

N#Cc1ccccc1Sc1ccc(C(F)(F)F)cc1N

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.64
CYP3A4 P08684 1/20 0.64
CYP2C9 P11712 1/20 0.64
CYP2C19 P33261 1/20 0.64
SLC6A2 P23975 2/20 0.56
SLC6A4 P31645 2/20 0.56
SLC6A3 Q01959 2/20 0.56
ALDH1A1 P00352 7/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
MAPT P10636 4/20 0.51
LMNA P02545 2/20 0.51
KDM4E B2RXH2 3/20 0.43
HPGD P15428 3/20 0.43
AR P10275 3/20 0.41
PGR P06401 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
GAA P10253 1/20 0.40
GFER P55789 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8881283 0.85 CYP1A2 (0.64) CYP1A2CYP3A4CYP2C9CYP2C19SLC6A2
SCHEMBL8879551 0.82 SLC6A2 (0.43) CYP1A2CYP3A4CYP2C9CYP2C19SLC6A2
SCHEMBL9316404 0.80 ALDH1A1 (0.57) CYP1A2CYP3A4CYP2C9CYP2C19SLC6A2
SCHEMBL1772241 0.79 CYP1A2 (1.00) CYP1A2CYP3A4CYP2C9CYP2C19SLC6A2
SCHEMBL11704957 0.76 SLC6A2 (0.56) SLC6A2SLC6A4SLC6A3ALDH1A1SMN1; SMN2
SCHEMBL11707664 0.76 KDM4E (0.60) CYP1A2CYP3A4CYP2C9CYP2C19SLC6A2
SCHEMBL463600 0.76 AR (0.47) ALDH1A1MAPTLMNAKDM4EHPGD
SCHEMBL8533879 0.75 SLC6A4 (0.70) SLC6A2SLC6A4SLC6A3MAPTLMNA
SCHEMBL8530833 0.75 SLC6A4 (0.70) SLC6A2SLC6A4SLC6A3MAPTLMNA
SCHEMBL100732 0.75 CYP1A2 (0.76) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607929-A Antiviral dibenzothiazepinone derivatives GLAXO WELLCOME INC. (US) 1997-03-04 US disclosed
US-5589474-A Dibenzothiazepinthione as antiviral agents GLAXO WELLCOME INC. (US) 1996-12-31 US disclosed
EP-0583288-A1 ANTIVIZAL DIBENZOTHIAZEPINONE DERIVATIVES THE WELLCOME FOUNDATION LIMITED (GB) 1994-02-23 EP disclosed
EP-0583317-A1 DIBENZOTHIAZEPINTHIONE AS ANTIVIRAL AGENTS THE WELLCOME FOUNDATION LIMITED (GB) 1994-02-23 EP disclosed
WO-1992019277-A1 ANTIVIRAL DIBENZOTHIAZEPINONE DERIVATIVES THE WELLCOME FOUNDATION LIMITED (GB) 1992-11-12 WO disclosed
WO-1992019607-A1 DIBENZOTHIAZEPINTHIONE AS ANTIVIRAL AGENTS THE WELLCOME FOUNDATION LIMITED (GB) 1992-11-12 WO disclosed