SCHEMBL8882797

SCHEMBL8882797

O=C1NCCC1(CCOC1CCCCO1)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 12/20 0.39
SLC6A3 Q01959 11/20 0.39
SLC6A2 P23975 10/20 0.39
PDE4A P27815 3/20 0.37
PDE4B Q07343 3/20 0.37
PDE4C Q08493 3/20 0.37
PDE4D Q08499 3/20 0.37
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
KDM4C Q9H3R0 1/20 0.34
CYP19A1 P11511 1/20 0.34
CYP3A4 P08684 2/20 0.33
TACR1 P25103 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRL1 P41146 1/20 0.33
SLC6A9 P48067 1/20 0.33
SLC6A5 Q9Y345 1/20 0.33
CYP1A1 P04798 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9027067 0.95 SLC6A4 (0.38) SLC6A4SLC6A3SLC6A2PDE4APDE4B
SCHEMBL8702363 0.89 MEN1 (0.37) SLC6A4SLC6A3SLC6A2PDE4APDE4B
SCHEMBL7935208 0.82 SLC6A2 (0.41) SLC6A4SLC6A3SLC6A2MEN1KMT2A
SCHEMBL4630541 0.78 SLC6A3 (0.37) SLC6A4SLC6A3SLC6A2MEN1KMT2A
SCHEMBL6950573 0.78 TACR1 (0.39) SLC6A4SLC6A3SLC6A2TACR1CYP2D6
SCHEMBL7765670 0.78 SLC6A3 (0.39) SLC6A4SLC6A3SLC6A2MEN1KMT2A
SCHEMBL7766689 0.78 SLC6A3 (0.39) SLC6A4SLC6A3SLC6A2TACR1CYP2D6
SCHEMBL6957304 0.78 SLC6A2 (0.50) SLC6A4SLC6A3SLC6A2CYP3A4CYP1A1
SCHEMBL7077339 0.77 SLC6A4 (0.57) SLC6A4SLC6A3SLC6A2CYP3A4CYP1A1
SCHEMBL8291781 0.77 SLC6A3 (0.46) SLC6A4SLC6A3SLC6A2KDM4CCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5607947-A Pyrrolidinyl tachykinin receptor antagonists ELI LILLY AND COMPANY (US) 1997-03-04 US disclosed
EP-0714891-A1 Heterocyclic tachykinin receptor antagonists ELI LILLY AND COMPANY (US) 1996-06-05 EP disclosed