SCHEMBL8883301

SCHEMBL8883301

CC(C)Oc1cc(C(=O)O)cnc1C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 3/20 0.49
RXRA P19793 3/20 0.45
KMT2A Q03164 1/20 0.43
RXRB P28702 2/20 0.40
RXRG P48443 1/20 0.40
GCK P35557 4/20 0.38
EP300 Q09472 2/20 0.38
RARA P10276 1/20 0.38
RARB P10826 1/20 0.38
RARG P13631 1/20 0.38
HCAR3 P49019 1/20 0.38
KCNQ3 O43525 1/20 0.38
KCNQ2 O43526 1/20 0.38
ALDH1A1 P00352 1/20 0.38
KMO O15229 1/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA3 P07451 1/20 0.37
PKM P14618 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8884248 0.84 CYP2C9 (0.51) XDHRXRAKMT2ARXRBRXRG
SCHEMBL976853 0.82 XDH (0.48) XDHRXRAKMT2ARXRBGCK
SCHEMBL8882930 0.82 RXRA (0.41) XDHRXRAKMT2ARXRBRXRG
SCHEMBL8768358 0.81 CA12 (0.53) CA12CA1CA2CA3PKM
SCHEMBL8875662 0.81 XDH (0.51) XDHRXRARXRBRXRGGCK
SCHEMBL7359867 0.80 XDH (0.46) XDHRXRAKMT2ARXRBRXRG
SCHEMBL8882657 0.78 XDH (0.53) XDHRXRAKMT2ARARBALDH1A1
SCHEMBL8881108 0.78 TSHR (0.53) RXRA
SCHEMBL1421009 0.78 PTGS2 (0.47) XDHKMT2ACA12CA1CA2
SCHEMBL8882488 0.75 RXRA (0.46) RXRAKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5658933-A Substituted heterocyclic carboxamide esters, their preparation and their use as pharmaceuticals HOECHST AKTIENGESELLSCHAFT (DE) 1997-08-19 US disclosed