SCHEMBL8883572

SCHEMBL8883572

CCOC(=O)c1cnc(C(=O)O)c(OCc2ccc(C(C)C)cc2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 2/20 0.48
RXRB P28702 1/20 0.48
MAOB P27338 4/20 0.47
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
P2RY12 Q9H244 2/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
MRGPRX4 Q96LA9 2/20 0.42
EGLN1 Q9GZT9 1/20 0.41
PPIA P62937 2/20 0.39
BRD4 O60885 1/20 0.39
GABRP O00591 1/20 0.39
GABRD O14764 1/20 0.39
GABRA1 P14867 1/20 0.39
GABRB1 P18505 1/20 0.39
GABRG2 P18507 1/20 0.39
GABRB3 P28472 1/20 0.39
GABRA5 P31644 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8890310 0.89 MRGPRX4 (0.52) MAOBP2RY12CYP2C9CYP2C19MRGPRX4
SCHEMBL8885039 0.88 RXRA (0.58) RXRARXRBNPC1RAB9AMRGPRX4
SCHEMBL8881676 0.87 PPIA (0.49) RXRARXRBMAOBNPC1RAB9A
SCHEMBL8885115 0.86 MAOB (0.54) RXRARXRBMAOBNPC1RAB9A
SCHEMBL8883579 0.86 MAOB (0.48) RXRARXRBMAOBL3MBTL1CYP2C9
SCHEMBL8883498 0.86 MAOB (0.48) RXRARXRBMAOBP2RY12CYP2C9
SCHEMBL8883630 0.85 RXRA (0.45) RXRARXRBNPC1RAB9AMRGPRX4
SCHEMBL8882407 0.83 MAOB (0.62) RXRARXRBMAOBCYP2C9CYP2C19
SCHEMBL8885505 0.83 RXRA (0.43) RXRARXRBNPC1RAB9AMRGPRX4
SCHEMBL8881837 0.83 MAOB (0.53) RXRARXRBMAOBCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5658933-A Substituted heterocyclic carboxamide esters, their preparation and their use as pharmaceuticals HOECHST AKTIENGESELLSCHAFT (DE) 1997-08-19 US disclosed