SCHEMBL8890310

SCHEMBL8890310

CCOC(=O)c1cnc(C(=O)O)c(OCc2ccc(Cl)cc2)c1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 2/20 0.52
MAOB P27338 4/20 0.48
XDH P47989 1/20 0.47
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
NR4A2 P43354 2/20 0.44
HDAC8 Q9BY41 2/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
TACR2 P21452 1/20 0.44
TDP1 Q9NUW8 1/20 0.43
POLB P06746 1/20 0.43
KMT2A Q03164 1/20 0.43
PPARA Q07869 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPK1 P28482 1/20 0.43
P2RY12 Q9H244 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8881676 0.89 PPIA (0.49) MRGPRX4MAOBCYP2C9CYP2C19KMT2A
SCHEMBL8883572 0.89 RXRA (0.48) MRGPRX4MAOBCYP2C9CYP2C19P2RY12
SCHEMBL8885115 0.88 MAOB (0.54) MRGPRX4MAOBCYP2C9CYP2C19TDP1
SCHEMBL8883579 0.88 MAOB (0.48) MRGPRX4MAOBXDHCYP2C9CYP2C19
SCHEMBL8883498 0.88 MAOB (0.48) MAOBXDHCYP2C9CYP2C19NR4A2
SCHEMBL8882346 0.87 MRGPRX4 (0.49) MRGPRX4XDHNR4A2ALDH1A1
SCHEMBL8884599 0.86 MRGPRX4 (0.60) MRGPRX4XDHNR4A2HDAC8HDAC1
SCHEMBL8882407 0.85 MAOB (0.62) MRGPRX4MAOBCYP2C9CYP2C19PPARA
SCHEMBL8881837 0.84 MAOB (0.53) MRGPRX4MAOBCYP2C9CYP2C19
SCHEMBL8881322 0.84 MAOB (0.48) MRGPRX4MAOBCYP2C9CYP2C19KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5658933-A Substituted heterocyclic carboxamide esters, their preparation and their use as pharmaceuticals HOECHST AKTIENGESELLSCHAFT (DE) 1997-08-19 US disclosed