SCHEMBL8885115

SCHEMBL8885115

CCOC(=O)c1cnc(C(=O)O)c(OCc2ccc(OCC)cc2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.54
RXRA P19793 1/20 0.47
RXRB P28702 1/20 0.47
SMN1; SMN2 Q16637 4/20 0.46
TP53 P04637 1/20 0.46
PKM P14618 1/20 0.46
NFKB1 P19838 1/20 0.46
NFKB2 Q00653 1/20 0.46
RELA Q04206 1/20 0.46
MRGPRX4 Q96LA9 1/20 0.46
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
NPC1 O15118 5/20 0.43
RAB9A P51151 5/20 0.43
MAPT P10636 2/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
GABRA1 P14867 2/20 0.42
GABRG2 P18507 2/20 0.42
GABRB3 P28472 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8881676 0.89 PPIA (0.49) MAOBRXRARXRBSMN1; SMN2MRGPRX4
SCHEMBL8881837 0.89 MAOB (0.53) MAOBRXRARXRBMRGPRX4CYP2C9
SCHEMBL8883579 0.88 MAOB (0.48) MAOBRXRARXRBMRGPRX4CYP2C9
SCHEMBL8890310 0.88 MRGPRX4 (0.52) MAOBMRGPRX4CYP2C9CYP2C19ALDH1A1
SCHEMBL8883498 0.88 MAOB (0.48) MAOBRXRARXRBCYP2C9CYP2C19
SCHEMBL8883572 0.86 RXRA (0.48) MAOBRXRARXRBMRGPRX4CYP2C9
SCHEMBL8882407 0.85 MAOB (0.62) MAOBRXRARXRBMRGPRX4CYP2C9
SCHEMBL8882705 0.85 CYP2C9 (0.56) MAOBCYP2C9CYP2C19NPC1RAB9A
SCHEMBL8881322 0.84 MAOB (0.48) MAOBSMN1; SMN2TP53MRGPRX4CYP2C9
SCHEMBL27404312 0.81 TSHR (0.52) RXRASMN1; SMN2MRGPRX4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5658933-A Substituted heterocyclic carboxamide esters, their preparation and their use as pharmaceuticals HOECHST AKTIENGESELLSCHAFT (DE) 1997-08-19 US disclosed