SCHEMBL8884367

SCHEMBL8884367

NCC(=O)NC(=O)c1nccc(OCC(F)(F)F)c1O

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
KDM4E B2RXH2 1/20 0.37
CNR2 P34972 4/20 0.37
GSK3B P49841 7/20 0.36
GSK3A P49840 5/20 0.36
ALDH1A1 P00352 5/20 0.36
MAPT P10636 1/20 0.36
MAPK1 P28482 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
LOXL2 Q9Y4K0 1/20 0.34
POLB P06746 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8881065 0.90 CNR2 (0.33) CYP1A2CYP2C9CNR2LOXL2
SCHEMBL8880853 0.88 CYP1A2 (0.31) CYP1A2CYP2C9MAPT
SCHEMBL8883329 0.88 KMT2A (0.42) CYP1A2CYP2C9KDM4EALDH1A1MAPT
SCHEMBL9254540 0.84 CYP1A2 (0.43) CYP1A2CYP2C9KDM4ECNR2GSK3B
SCHEMBL8884727 0.84 MAOB (0.44) ALDH1A1
SCHEMBL8883715 0.83 SMN1; SMN2 (0.37) KDM4EALDH1A1SMN1; SMN2POLB
SCHEMBL8882392 0.83 ALDH1A1 (0.39) ALDH1A1MAPT
SCHEMBL8883675 0.82 GSK3B (0.42) CYP1A2CYP2C9KDM4ECNR2GSK3B
SCHEMBL8884435 0.82 TDP1 (0.42) CYP1A2KDM4EMAPTMAPK1SMN1; SMN2
SCHEMBL8882459 0.81 IKBKB (0.39) KDM4EALDH1A1MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5620995-A Substituted heterocyclic carboxyamides, their preparation and their use as pharmaceuticals HOECHST AKTIENGESELLSCHAFT (DE) 1997-04-15 US disclosed