SCHEMBL9254540

SCHEMBL9254540

COc1c(OCC(F)(F)F)ccnc1C(=O)NC(=O)CN

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
ALDH1A1 P00352 1/20 0.37
GSK3B P49841 7/20 0.36
MAPT P10636 2/20 0.36
S1PR1 P21453 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
KDM4E B2RXH2 1/20 0.35
CNR2 P34972 1/20 0.35
GSK3A P49840 5/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34
CYP17A1 P05093 1/20 0.34
BACE1 P56817 1/20 0.34
BACE2 Q9Y5Z0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8884367 0.84 CYP1A2 (0.40) CYP1A2CYP2C9ALDH1A1GSK3BMAPT
SCHEMBL8786684 0.82 CYP1A2 (0.39) CYP1A2CYP2C9ALDH1A1GSK3BMAPT
SCHEMBL8881151 0.80 L3MBTL1 (0.41) CYP1A2CYP2C9ALDH1A1GSK3BMAPT
SCHEMBL8884435 0.76 TDP1 (0.42) CYP1A2MAPTTDP1KDM4ECYP2C19
SCHEMBL8881065 0.75 CNR2 (0.33) CYP1A2CYP2C9CNR2
SCHEMBL8880853 0.74 CYP1A2 (0.31) CYP1A2CYP2C9MAPT
SCHEMBL8883329 0.74 KMT2A (0.42) CYP1A2CYP2C9ALDH1A1MAPTTDP1
SCHEMBL8786282 0.73 CARM1 (0.33) CYP1A2CYP2C9
SCHEMBL8779238 0.71 CYP1A2 (0.36) CYP1A2CYP2C9ALDH1A1GSK3BMAPT
SCHEMBL8883715 0.70 SMN1; SMN2 (0.37) ALDH1A1TDP1KDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-7228571-A None JP disclosed
JP-H07228571-A SUBSTITUTED HETEROCYCLIC CARBOXAMIDES, THEIR PRODUCTION AND THEIR USE AS PHARMACEUTICALS HOECHST AG 1995-08-29 JP disclosed