SCHEMBL8886431

SCHEMBL8886431

CCC(C)C1COC(C(C)C)C(=O)N1C(=O)OC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NR1H3 Q13133 2/20 0.36
NR1H2 P55055 1/20 0.36
PLA2G10 O15496 1/20 0.35
PLA2G5 P39877 1/20 0.35
KLK7 P49862 6/20 0.33
KLK5 Q9Y337 5/20 0.33
GPR119 Q8TDV5 2/20 0.31
CHRM2 P08172 1/20 0.31
CHRM1 P11229 1/20 0.31
CHRM3 P20309 1/20 0.31
SPHK1 Q9NYA1 1/20 0.30
GRIN2B Q13224 1/20 0.30
GRIN2C Q14957 1/20 0.30
PRSS1 P07477 2/20 0.30
PRSS2 P07478 2/20 0.30
PRSS3 P35030 2/20 0.30
KDM4E B2RXH2 1/20 0.30
MAPT P10636 1/20 0.30
THRB P10828 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8073190 1.00 NR1H3 (0.36) NR1H3NR1H2PLA2G10PLA2G5KLK7
SCHEMBL8078090 0.85 KLK7 (0.39) NR1H3NR1H2KLK7KLK5GPR119
SCHEMBL8065148 0.84 NR1H3 (0.36) NR1H3NR1H2PLA2G10PLA2G5KLK7
SCHEMBL8885982 0.81 NR1H3 (0.34) NR1H3NR1H2PLA2G10PLA2G5KLK7
SCHEMBL8065492 0.81 NR1H3 (0.34) NR1H3NR1H2PLA2G10PLA2G5KLK7
SCHEMBL8073393 0.81 NR1H3 (0.34) NR1H3NR1H2PLA2G10PLA2G5KLK7
SCHEMBL8886010 0.78 KLK7 (0.48) NR1H3NR1H2PLA2G10PLA2G5KLK7
SCHEMBL5891618 0.78 KLK7 (0.48) NR1H3NR1H2PLA2G10PLA2G5KLK7
SCHEMBL8884829 0.78 KLK7 (0.48) NR1H3NR1H2PLA2G10PLA2G5KLK7
SCHEMBL5891823 0.78 GLA (0.39) NR1H3NR1H2PLA2G10PLA2G5KLK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5686472-A ANTICARCINOGENIC AND -TUMOR AGENTS; SIDE EFFECT REDUCTION; INHIBITION OF FARNESYLATION OF THE RAS PROTEIN MERCK & CO., INC. (US) 1997-11-11 US disclosed