SCHEMBL8887662

SCHEMBL8887662

COc1ccc2c(c1)CCCC2CCNC(=O)C(C)C

nearest known ligand 0.72

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 15/20 0.72
MTNR1B P49286 14/20 0.72
NQO2 P16083 13/20 0.72
TRPV1 Q8NER1 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8887708 0.93 MTNR1A (0.83) MTNR1AMTNR1BNQO2
SCHEMBL7956485 0.91 MTNR1A (0.87) MTNR1AMTNR1BNQO2TRPV1
SCHEMBL8886502 0.85 MTNR1A (0.62) MTNR1AMTNR1BNQO2TRPV1
SCHEMBL8885947 0.84 MTNR1A (0.67) MTNR1AMTNR1BNQO2TRPV1
SCHEMBL7956487 0.84 MTNR1A (1.00) MTNR1AMTNR1BNQO2
SCHEMBL7943739 0.84 MTNR1A (1.00) MTNR1AMTNR1BNQO2
SCHEMBL8887067 0.83 MTNR1A (0.73) MTNR1AMTNR1BNQO2TRPV1
SCHEMBL10175563 0.83 MTNR1A (0.60) MTNR1AMTNR1BNQO2TRPV1
SCHEMBL8886469 0.80 MTNR1A (0.82) MTNR1AMTNR1BNQO2
SCHEMBL5172930 0.79 SIGMAR1 (0.61)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5661186-A MELATONERGIC EFFECT; CENTRAL NERVOUS SYSTEM DISODERS BRISTOL-MYERS SQUIBB CO. (US) 1997-08-26 US claimed
EP-0728738-A1 Tetralinyl- and indanyl-ethylamides having melatonergic activity BRISTOL-MYERS SQUIBB COMPANY (US) 1996-08-28 EP claimed