SCHEMBL8887683

SCHEMBL8887683

Cc1nn(COC(C)[Si](C)(C)C)c2cc(O)ccc12

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.39
KMO O15229 1/20 0.37
SLC22A12 Q96S37 10/20 0.36
ADORA2A P29274 2/20 0.36
ADORA2B P29275 2/20 0.36
HTR1A P08908 2/20 0.34
ADRA2A P08913 2/20 0.34
ADRA2B P18089 2/20 0.34
ADRA2C P18825 2/20 0.34
HTR2A P28223 2/20 0.34
HTR2C P28335 2/20 0.34
HTR2B P41595 2/20 0.34
HTR1D P28221 1/20 0.34
HTR7 P34969 1/20 0.34
HTR4 Q13639 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8889173 0.78 ADORA2A (0.41) ADORA2AADORA2B
SCHEMBL3562422 0.76 ADORA2A (0.36) ADORA2AADORA2BHTR2AHTR2C
SCHEMBL18853871 0.75 ESR1 (0.63) ESR1KMOSLC22A12ADORA2AADORA2B
SCHEMBL3136016 0.75 HTR2A (0.56) ESR1KMOSLC22A12ADORA2AADORA2B
SCHEMBL8887595 0.71 ESR1 (0.36) ESR1
SCHEMBL6486543 0.70 KMO (0.36) KMOADORA2A
SCHEMBL177096 0.70 SLC22A12 (0.51) SLC22A12
SCHEMBL15723742 0.69 GRM4 (0.43) ESR1HTR1AADRA2AADRA2BADRA2C
Fumaric Acid SCHEMBL4845606 0.68 HTR2A (0.47) ESR1KMOSLC22A12HTR1AADRA2A
Fumaric Acid SCHEMBL4845619 0.68 HTR2A (0.47) ESR1KMOSLC22A12HTR1AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5631264-A NEUROLOGICAL DISORDERS SANOFI WINTHROP, INC. (US) 1997-05-20 US disclosed
US-5554620-A Substituted 6,11-ethano-6,11-dihydrobenzo[b] quinolizinium salts and compositions and methods of use thereof STERLING WINTHROP INC. (US) 1996-09-10 US disclosed
EP-0656359-A1 Substituted 6,11-ethano-6,11-dihydrobenzo[b]quinolizinium salts and compositionsand methods of use thereof STERLING WINTHROP INC. (US) 1995-06-07 EP disclosed