SCHEMBL8889173

SCHEMBL8889173

Cc1nn(COC(C)[Si](C)(C)C)c2cc(Br)c(Br)cc12

nearest known ligand 0.41

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.41
ADORA2B P29275 4/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3562422 0.84 ADORA2A (0.36) ADORA2AADORA2B
SCHEMBL8887683 0.78 ESR1 (0.39) ADORA2AADORA2B
SCHEMBL8889178 0.75 ADORA2A (0.41) ADORA2AADORA2B
SCHEMBL3628566 0.68
SCHEMBL6486543 0.67 KMO (0.36) ADORA2A
SCHEMBL8226285 0.66 DGAT1 (0.40) ADORA2AADORA2B
SCHEMBL9232701 0.64 HTR2A (0.35)
SCHEMBL14561774 0.62 ADORA2A (0.36) ADORA2AADORA2B
SCHEMBL26912128 0.61
SCHEMBL11976878 0.59 DGAT1 (0.43) ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5631264-A NEUROLOGICAL DISORDERS SANOFI WINTHROP, INC. (US) 1997-05-20 US disclosed
US-5554620-A Substituted 6,11-ethano-6,11-dihydrobenzo[b] quinolizinium salts and compositions and methods of use thereof STERLING WINTHROP INC. (US) 1996-09-10 US disclosed