SCHEMBL8887703

SCHEMBL8887703

N#CNc1cc(NC#N)cc(C(=O)O)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 6/20 0.42
KMT2A Q03164 6/20 0.42
POLB P06746 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
PKM P14618 1/20 0.41
CA12 O43570 2/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA7 P43166 2/20 0.39
CA9 Q16790 2/20 0.39
CA14 Q9ULX7 2/20 0.39
TPMT P51580 3/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
CA3 P07451 1/20 0.38
MAPT P10636 1/20 0.38
SELL P14151 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18095930 0.96 PKM (0.46) MEN1KMT2APOLBL3MBTL1PKM
SCHEMBL20010428 0.81 PKM (0.36) MEN1KMT2APOLBL3MBTL1PKM
Water SCHEMBL8887299 0.80 AKR1C3 (0.51) MEN1KMT2APOLBL3MBTL1PKM
SCHEMBL2346165 0.80 AKR1C3 (0.51) MEN1KMT2APOLBL3MBTL1PKM
SCHEMBL7287581 0.78 TSHR (0.52) MEN1KMT2ACA12CA1CA2
SCHEMBL9726925 0.76 PKM (0.47) MEN1KMT2APOLBL3MBTL1PKM
SCHEMBL11737816 0.71 KDM5A (0.48) MEN1KMT2APOLBL3MBTL1PKM
SCHEMBL10665479 0.71 AKR1C3 (0.35) MEN1KMT2APOLBKDM4EMAPT
SCHEMBL2884556 0.70 KDM4E (0.61) MEN1KMT2APOLBL3MBTL1PKM
SCHEMBL999842 0.70 CYP1A2 (0.47) MEN1KMT2APOLBL3MBTL1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5602277-A Substituted benzene derivatives useful as neuraminidase inhibitors BIOCRYST PHARMACEUTICALS, INC. (US) 1997-02-11 US disclosed
WO-1996030329-A1 SUBSTITUTED BENZENE DERIVATIVES USEFUL AS NEURAMINIDASE INHIBITORS BIOCRYST PHARMACEUTICALS, INCORPORATED (US) 1996-10-03 WO disclosed